Guanfacine hydrochloride

Catalog No.: A15098

α2A-adrenoceptor agonist

Guanfacine hydrochloride

Guanfacine hydrochloride Chemical Structure

CAS NO. 29110-48-3

Guanfacine hydrochloride, an anti-hypertensive agent, is a selective α2A-adrenoceptor agonist with Kd of 31 nM and displays 60-fold selectivity over α2B-adrenoceptors.

Availability: In stock

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10 mg
$50.00
50 mg
$150.00
100 mg
$290.00
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Biological Activity

Guanfacine hydrochloride, an anti-hypertensive agent, is a selective α2A-adrenoceptor agonist with Kd of 31 nM and displays 60-fold selectivity over α2B-adrenoceptors.
Targets
α2A-adrenoceptor
In vitro DMSO 48 mg/mL (169.88 mM)
Water 26 mg/mL (92.01 mM)
Ethanol 48 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 35.39 mL 176.96 mL 353.92 mL
0.5 mM 7.08 mL 35.39 mL 70.78 mL
1 mM 3.54 mL 17.7 mL 35.39 mL
5 mM 0.71 mL 3.54 mL 7.08 mL

*The above data is based on the productmolecular weight 282.55. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15098
Actions Agonist
CAS No. 29110-48-3
Formula C9H10Cl3N3O
M. Wt 282.55
Purity >98%
Synonyms Guanfacine, Tenex, Intuniv
SMILES C1=CC(=C(C(=C1)Cl)CC(=O)N=C(N)N)Cl.Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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