GW679769 (Casopitant)

Catalog No.: A13103

NK1 receptor antagonist

GW679769 (Casopitant)

GW679769 (Casopitant) Chemical Structure

CAS NO. 414910-27-3 (free base), 414910-30-8 (mesylate)

Casopitant mesylate is the mesylate salt of a centrally-acting neurokinin 1 (NK1) receptor antagonist with antidepressant and antiemetic activities.

Availability: In stock

Package Price Qty
5 mg
$350.00
10 mg
$600.00
25 mg
$1,200.00
50 mg
$2,000.00
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Biological Activity

Casopitant mesylate is the mesylate salt of a centrally-acting neurokinin 1 (NK1) receptor antagonist with antidepressant and antiemetic activities.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.22 mL 81.09 mL 162.18 mL
0.5 mM 3.24 mL 16.22 mL 32.44 mL
1 mM 1.62 mL 8.11 mL 16.22 mL
5 mM 0.32 mL 1.62 mL 3.24 mL

*The above data is based on the productmolecular weight 616.61. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13103
Actions Antagonist
CAS No. 414910-27-3 (free base), 414910-30-8 (mesylate)
Formula C30H35F7N4O2
M. Wt 616.61
Purity >98%
Synonyms GW 679769, GW-679769
SMILES CC1=C(C=CC(=C1)F)[[email protected]]2C[[email protected]](CCN2C(=O)N(C)[[email protected]](C)C3=CC(=CC(=C3)C(F)(F)F)C(F)(F)F)N4CCN(CC4)C(=O)C
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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