GW791343 trihydrochloride

Catalog No.: A21204

P2X7 allosteric modulator

GW791343 trihydrochloride

GW791343 trihydrochloride Chemical Structure

CAS NO. 309712-55-8

GW791343 3Hcl is a P2X7 allosteric modulator; exhibits species-specific activity and acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2).

Availability: In stock

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1 mg

Regular Price: $320.00

Special Price $256.00

5 mg

Regular Price: $960.00

Special Price $768.00

10 mg

Regular Price: $1,600.00

Special Price $1,280.00

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Biological Activity

GW791343 3Hcl is a P2X7 allosteric modulator; exhibits species-specific activity and acts as a negative allosteric modulator of human P2X7 (pIC50 = 6.9 - 7.2).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.67 mL 103.35 mL 206.69 mL
0.5 mM 4.13 mL 20.67 mL 41.34 mL
1 mM 2.07 mL 10.33 mL 20.67 mL
5 mM 0.41 mL 2.07 mL 4.13 mL

*The above data is based on the productmolecular weight 483.81. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21204
Actions Modulator
CAS No. 309712-55-8
Formula C20H27Cl3F2N4O
M. Wt 483.81
Purity >98%
Synonyms GW 791343, GW-791343
SMILES O=C(NC1=CC(CN2CCNCC2)=CC=C1C)CNC3=CC=C(F)C(F)=C3.[H]Cl.[H]Cl.[H]Cl
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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