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GW9662-d5

Stable Isotope

GW9662-d5 is a deuterium-labeled derivative of the potent PPARγ antagonist GW9662. It exhibits an IC50 of 3.3 nM for PPARγ, demonstrating significant selectivity with 10-fold affinity over PPARα and 1000-fold over PPARδ. This stable isotope variant is ideal for tracer studies and applications in metabolic research, particularly in understanding the role of PPARγ in insulin sensitivity and adipogenesis.

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Specifications

Manufacturer	Adooq Bioscience
CAS Number	2117730-84-2
Applications	Stable Isotope
Formula	C₁₃H₄D₅ClN₂O₃
Molecular Weight	281.71
SMILES	ClC1=CC=C(C=C1C(NC2=C(C([2H])=C(C([2H])=C2[2H])[2H])[2H])=O)[N+]([O-])=O

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.