GW9662-d5 is a deuterium-labeled derivative of the potent PPARγ antagonist GW9662. It exhibits an IC50 of 3.3 nM for PPARγ, demonstrating significant selectivity with 10-fold affinity over PPARα and 1000-fold over PPARδ. This stable isotope variant is ideal for tracer studies and applications in metabolic research, particularly in understanding the role of PPARγ in insulin sensitivity and adipogenesis.
GW9662-d5 is a deuterium-labeled derivative of the potent PPARγ antagonist GW9662. It exhibits an IC50 of 3.3 nM for PPARγ, demonstrating significant selectivity with 10-fold affinity over PPARα and 1000-fold over PPARδ. This stable isotope variant is ideal for tracer studies and applications in metabolic research, particularly in understanding the role of PPARγ in insulin sensitivity and adipogenesis.
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