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Biological Activity
HTH-01-015 is a potent and selective inhibitor of NUAK1 (IC50 = 100 nM) and does not affect the activity of a panel of 139 other kinases, including additional AMPK family members.
Targets
| NUAK1 | NUAK2 | |||
| 100 nM | >10 μM |
| In vitro | DMSO | Warmed: 54 mg/mL (115.24 mM) | |
| Water | Insoluble | ||
| Ethanol | 28 mg/mL (59.75 mM) | ||
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 21.34 mL | 106.71 mL | 213.42 mL |
| 0.5 mM | 4.27 mL | 21.34 mL | 42.68 mL |
| 1 mM | 2.13 mL | 10.67 mL | 21.34 mL |
| 5 mM | 0.43 mL | 2.13 mL | 4.27 mL |
*The above data is based on the productmolecular weight 468.56. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A16281 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1613724-42-7 |
| Formula | C26H28N8O |
| M. Wt | 468.56 |
| Purity | >98% |
| Synonyms | HTH01-015, HTH 01-015 |
| SMILES | CC1=C(N(C)C(C2=CC(C=CC=C3)=C3C=C2N4C)=O)C4=NC(NC5=CN(N=C5)C6CCNCC6)=N1 |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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