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HTH-01-015

Catalog No.: A16281

NUAK1 inhibitor

HTH-01-015

HTH-01-015 Chemical Structure

CAS NO. 1613724-42-7

HTH-01-015 is a potent and selective inhibitor of NUAK1 (IC50 = 100 nM) and does not affect the activity of a panel of 139 other kinases, including additional AMPK family members.

Availability: In stock

Package Price Qty
5 mg
$90.00
10 mg
$120.00
50 mg
$400.00
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Biological Activity

HTH-01-015 is a potent and selective inhibitor of NUAK1 (IC50 = 100 nM) and does not affect the activity of a panel of 139 other kinases, including additional AMPK family members.
Targets
NUAK1 NUAK2
100 nM>10 μM
In vitro DMSO Warmed: 54 mg/mL (115.24 mM)
Water Insoluble
Ethanol 28 mg/mL (59.75 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 21.34 mL 106.71 mL 213.42 mL
0.5 mM 4.27 mL 21.34 mL 42.68 mL
1 mM 2.13 mL 10.67 mL 21.34 mL
5 mM 0.43 mL 2.13 mL 4.27 mL

*The above data is based on the productmolecular weight 468.56. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16281
Actions Inhibitor
CAS No. 1613724-42-7
Formula C26H28N8O
M. Wt 468.56
Purity >98%
Synonyms HTH01-015, HTH 01-015
SMILES CC1=C(N(C)C(C2=CC(C=CC=C3)=C3C=C2N4C)=O)C4=NC(NC5=CN(N=C5)C6CCNCC6)=N1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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