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CDK inhibitor

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Catalog No. A11220

Availability:Stock in USAIn stock Shipped in 7-10 Days

Product Name Catalog No. Price Qty
Kenpaullone 10mg A11220-10

Regular Price: $90.00

Special Price: $81.00

Kenpaullone 50mg A11220-50

Regular Price: $380.00

Special Price: $342.00

Kenpaullone 100mg A11220-100

Regular Price: $650.00

Special Price: $585.00

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Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

Kenpaullone is a potent inhibitor of CDK1/cyclin B (IC₅₀ = 400 nM), CDK2/cyclin A (IC₅₀ = 680nM) , CDK5 (IC₅₀ = 850nM) and with much less effect other kinases.


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Chemical Information

Catalog Num A11220
Actions Inhibitor
M. Wt 327.2
Formula C16H11BrN2O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 142273-20-9
Synonyms N/A

Biological Activity

Kenpaullone is a potent inhibitor of CDK1/cyclin B (IC₅₀ = 400 nM), CDK2/cyclin A (IC₅₀ = 680nM) , CDK5 (IC₅₀ = 850nM) and with much less effect other kinases.
Target Value
GSK-3βIC50: 0.23μM
CDK1/CyclinBIC50: 0.4μM
CDK2/CyclinAIC50: 0.68μM
CDK5/p35IC50: 0.85μM
CDK2/CyclinEIC50: 7.5μM
ERK2IC50: 9μM
c-SrcIC50: 15μM
CaseinKinase2IC50: 20μM
ERK1IC50: 20μM

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 30.56 mL 152.81 mL 305.62mL
0.5 mM 6.11 mL 30.56 mL 61.12 mL
1 mM 3.06 mL 15.28 mL 30.56 mL
5 mM 0.61 mL 3.06 mL 6.11 mL

*The above data is based on the productmolecular weight 327.2. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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