Ki16198

Catalog No.: A11966

LPA Receptor antagonist

Ki16198

Ki16198 Chemical Structure

CAS NO. 355025-13-7

Ki16198 is a potent LPA receptor antagonist and inhibits LPA1- and LPA3-induced inositol phosphate production with Ki of 0.34 μM and 0.93 μM, respectively.

Availability: In stock

Package Price Qty
5 mg
$160.00
10 mg
$259.00
25 mg
$500.00
50 mg
$749.00
10mM * 1mL in DMSO
$215.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Ki16198 is a potent LPA receptor antagonist and inhibits LPA1- and LPA3-induced inositol phosphate production with Ki of 0.34 μM and 0.93 μM, respectively.
Targets
LPA1 LPA3
0.34 μM(Ki)0.93 μM(Ki)
In vitro (25°C) DMSO 96 mg/mL (196.32 mM)
Water 96 mg/mL (196.32 mM)
Ethanol 35 mg/mL (71.57 mM)
In vivo 1% DMSO/30% polyethylene glycol/1% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.45 mL 102.25 mL 204.51 mL
0.5 mM 4.09 mL 20.45 mL 40.9 mL
1 mM 2.05 mL 10.23 mL 20.45 mL
5 mM 0.41 mL 2.05 mL 4.09 mL

*The above data is based on the productmolecular weight 488.98. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11966
Actions Antagonist
M. Wt 488.98
Formula C24H25ClN2O5S
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 355025-13-7
Synonyms Ki-16198
SMILES CC1=NOC(=C1NC(=O)OC(C)C2=CC=CC=C2Cl)C3=CC=C(C=C3)CSCCC(=O)OC

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