Ki16425

Name: Ki16425
SKU: A10501
Price: 30 USD
Rating: 5 (5 reviews)

Catalog No.: A10501

LPA Receptor Antagonist

Adooq's Ki16425 has been cited by 5 publications

Ki16425 is a LPA receptor antagonist with selectivity for LPA1 and LPA3 and exhibits Ki values of 0.34, 6.5, and 0.93 μM for the human LPA1, LPA2, and LPA3 receptors, respectively.

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Grouped product items
Size	Price	Stock
2mg	$30.00	In stock
5mg	$45.00	In stock
10mg	$85.00	In stock
25mg	$190.00	In stock
50mg	$355.00	In stock
100mg	$445.00	In stock
*10mM 1mL in DMSO**	$45.00	In stock
Bulk Size	Bulk Discount

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Important Notice: For research use only. We do not sell to patients.

Data Sheet

SDS

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Adooq Products cited in reputable paper

Adooq's Ki16425 has been cited by 5 publications

Maria F Fernandes, .et al. , Int J Mol Sci, 2022, Apr 9;23(8):4163 PMID: 35456981

Rieko Suenaga, .et al. , PLoS One, 2022, Feb 3;17(2):e0263296 PMID: 35113924

Inoue A, .et al. , Cell, 2019, Jun 13;177(7):1933-1947 PMID: 31160049

Taniguchi R, .et al. , Nature, 2017, Aug 17;548(7667):356-360 PMID: 28792932

T. HASHIMOTO, .et al. , Br J Dermatol., 2015, Nov;173(5):1334-6 PMID: 26122943

Biological Activity

Discription	Ki16425 is a LPA receptor antagonist with selectivity for LPA1 and LPA3 and exhibits Ki values of 0.34, 6.5, and 0.93 μM for the human LPA1, LPA2, and LPA3 receptors, respectively.

Product Information

Catalog Num	A10501
Formula	C23H23ClN2O5S
Molecular Weight	475
CAS Number	355025-24-0
SMILES	CC1=NOC(=C1NC(=O)OC(C)C2=CC=CC=C2Cl)C3=CC=C(C=C3)CSCCC(=O)O
Synonyms	Ki-16425
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 1 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility

In vitro (25°C)	DMSO	85 mg/mL (178.96 mM)
	Water	Insoluble
	Ethanol	85 mg/mL (178.96 mM)
In vivo	5% DMSO+95% Corn oil	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	21.05 mL	105.26 mL	210.53 mL
0.5 mM	4.21 mL	21.05 mL	42.11 mL
1 mM	2.11 mL	10.53 mL	21.05 mL
5 mM	0.42 mL	2.11 mL	4.21 mL

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