Fig. 1 · Structure
Documents & Downloads
KSQ-4279 (gentisate)
USP1/PARP1 Inhibitor
KSQ-4279 (gentisate) is a potent inhibitor of USP1 and selectively targets PARP1. This compound demonstrates significant potential in cancer research, showcasing its ability to disrupt key pathways involved in tumor progression and repair mechanisms. Its unique inhibitory properties make it a valuable tool for studying the molecular underpinnings of various cancer types and developing targeted therapeutic strategies.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Inhibitor |
| CAS Number | 2938991-80-9 |
| Applications | USP1/PARP1 Inhibitor |
| Formula | C34H31F3N8O5 |
| Molecular Weight | 688.66 |
| SMILES | O=C(C1=CC(O)=CC=C1O)O.FC(F)(C2=CN(C(C)C)C(C3=CC=C(CN4N=CC5=C4N=C(C6=C(C7CC7)N=CN=C6OC)N=C5)C=C3)=N2)F |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.