L-803087 is a highly potent and selective agonist of the somatostatin sst4 receptor, exhibiting a Ki value of 0.7 nM, which demonstrates over 280-fold selectivity compared to other somatostatin receptors. This compound is known to enhance AMPA-mediated hippocampal synaptic responses in vitro and has been shown to increase kainate-induced seizures in murine models. L-803087 is a valuable tool for investigating the pharmacological roles of sst4 receptors in neurological research.
L-803087 is a highly potent and selective agonist of the somatostatin sst4 receptor, exhibiting a Ki value of 0.7 nM, which demonstrates over 280-fold selectivity compared to other somatostatin receptors. This compound is known to enhance AMPA-mediated hippocampal synaptic responses in vitro and has been shown to increase kainate-induced seizures in murine models. L-803087 is a valuable tool for investigating the pharmacological roles of sst4 receptors in neurological research.
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