LB42708

Catalog No.: A14020

FTase inhibitor

LB42708

LB42708 Chemical Structure

CAS NO. 226929-39-1

LB42708 is a potent, orally active and selective nonpeptidic farnesyltransferase inhibitor (FTase inhibitor).

Availability: In stock

Package Price Qty
5 mg

Regular Price: $60.00

Special Price $54.00

10 mg

Regular Price: $100.00

Special Price $90.00

25 mg

Regular Price: $200.00

Special Price $180.00

10mM * 1mL in DMSO

Regular Price: $126.00

Special Price $113.40

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

LB42708 is a potent, orally active and selective nonpeptidic farnesyltransferase inhibitor (FTase inhibitor).
Targets
FTase (H-ras) FTase (N-ras) FTase (K-Ras)
0.8 nM1.2 nM2.0 nM
In vitro DMSO 100 mg/mL (180.03 mM)
Water <1 mg/mL (<1 mM)
Ethanol 86 mg/mL heating (154.82 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18 mL 90.02 mL 180.03 mL
0.5 mM 3.6 mL 18 mL 36.01 mL
1 mM 1.8 mL 9 mL 18 mL
5 mM 0.36 mL 1.8 mL 3.6 mL

*The above data is based on the productmolecular weight 555.46. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A14020
Actions Inhibitor
M. Wt 555.46
Formula C30H27BrN4O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 226929-39-1
Synonyms LB-42708, LB 42708
SMILES C1COCCN1C(=O)C2=CN(C=C2C3=CC=CC4=CC=CC=C43)CC5=CN=CN5CC6=CC=C(C=C6)Br

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