LEI-101 is a selective, orally bioavailable agonist of the cannabinoid CB2 receptor, exhibiting a pEC50 of 8 for human CB2. With a pKi of less than 4 for hERG, it demonstrates minimal off-target activity. This compound is approximately 100-fold more potent in binding to CB2 receptors compared to CB1 receptors, making it a valuable tool for research in pain modulation, inflammation, and neuroprotection studies.
LEI-101 is a selective, orally bioavailable agonist of the cannabinoid CB2 receptor, exhibiting a pEC50 of 8 for human CB2. With a pKi of less than 4 for hERG, it demonstrates minimal off-target activity. This compound is approximately 100-fold more potent in binding to CB2 receptors compared to CB1 receptors, making it a valuable tool for research in pain modulation, inflammation, and neuroprotection studies.
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