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Biological Activity
Linagliptin is a DPP-4 inhibitor, an enzyme that degrades the incretin hormones glucagon-like peptide-1 (GLP-1) and glucose-dependent insulinotropic polypeptide (GIP).
Targets
| DPP-4 | ||||
| 1 nM |
| In vitro (25°C) | DMSO | 16 mg/mL (33.85 mM) | |
| Water | Insoluble | ||
| Ethanol | 1 mg/mL (2.11 mM) | ||
| In vivo | 0.5% hydroxyethyl cellulose | 28 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 21.16 mL | 105.82 mL | 211.64 mL |
| 0.5 mM | 4.23 mL | 21.16 mL | 42.33 mL |
| 1 mM | 2.12 mL | 10.58 mL | 21.16 mL |
| 5 mM | 0.42 mL | 2.12 mL | 4.23 mL |
*The above data is based on the productmolecular weight 472.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A11224 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 668270-12-0 |
| Formula | C25H28N8O2 |
| M. Wt | 472.5 |
| Purity | >98% |
| Synonyms | BI-1356,Tradjenta,Trajenta |
| SMILES | CC#CCN1C2=C(N=C1N3CCC[C@H](C3)N)N(C(=O)N(C2=O)CC4=NC5=CC=CC=C5C(=N4)C)C |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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