LX-039 is a potent and selective estrogen receptor degrader with an EC50 value of 2.29 nM. Featuring an indole C-3 chlorine substituent, LX-039 demonstrates favorable pharmacokinetics in mouse models, characterized by low clearance and high maximum concentration (Cmax) following oral administration. Its efficacy in degrading estrogen receptors highlights its potential for anti-tumor applications in research settings.
LX-039 is a potent and selective estrogen receptor degrader with an EC50 value of 2.29 nM. Featuring an indole C-3 chlorine substituent, LX-039 demonstrates favorable pharmacokinetics in mouse models, characterized by low clearance and high maximum concentration (Cmax) following oral administration. Its efficacy in degrading estrogen receptors highlights its potential for anti-tumor applications in research settings.
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