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TGFβR-I Inhibitor

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Catalog No. A13446

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
LY364947 10mg A13446-10

Regular Price: $60.00

Special Price: $54.00

LY364947 25mg A13446-25

Regular Price: $120.00

Special Price: $108.00

LY364947 50mg A13446-50

Regular Price: $200.00

Special Price: $180.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

LY364947 is a diheteroaryl-substituted pyrazole compound used as a selective, ATP-competitive inhibitor of TGF-βRI (TGF-β Receptor I kinase).


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Chemical Information

Catalog Num A13446
Actions Inhibitor
M. Wt 272.3
Formula C17H12N4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 396129-53-6
Synonyms HTS 466284 ,TGF-β RI Kinase Inhibitor

Biological Activity

LY364947 is a diheteroaryl-substituted pyrazole compound used as a selective, ATP-competitive inhibitor of TGF-βRI (TGF-β Receptor I kinase).
TGFβRI (Cell-free assay) RIPK2 (Cell-free assay) CK1δ (Cell-free assay) TGFβRII (Cell-free assay) MLK-7K (Cell-free assay)
59 nM0.11 μM0.22 μM0.4 μM1.4 μM

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 36.72 mL 183.62 mL 367.24mL
0.5 mM 7.34 mL 36.72 mL 73.45 mL
1 mM 3.67 mL 18.36 mL 36.72 mL
5 mM 0.73 mL 3.67 mL 7.34 mL

*The above data is based on the productmolecular weight 272.3. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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