Mavatrep

Catalog No.: A15778

TRPV1 antagonist

Mavatrep

Mavatrep Chemical Structure

CAS NO. 956274-94-5

Mavatrep is an orally bioavailable TRPV1 antagonist (Ki=6.5 nM), exhibits minimal effect on the enzymatic activity (IC50 > 25 μM) of CYP isoforms 3A4, 1A2, and 2D6.

Availability: Out of stock

Package Price
2 mg
$180.00
5 mg
$350.00
10 mg
$500.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

Mavatrep is an orally bioavailable TRPV1 antagonist (Ki=6.5 nM), exhibits minimal effect on the enzymatic activity (IC50 > 25 μM) of CYP isoforms 3A4, 1A2, and 2D6.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.67 mL 118.36 mL 236.72 mL
0.5 mM 4.73 mL 23.67 mL 47.34 mL
1 mM 2.37 mL 11.84 mL 23.67 mL
5 mM 0.47 mL 2.37 mL 4.73 mL

*The above data is based on the productmolecular weight 422.44. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15778
Actions Antagonist
CAS No. 956274-94-5
Formula C25H21F3N2O
M. Wt 422.44
Purity >98%
Synonyms JNJ-39439335
SMILES CC(C)(C1=CC=CC=C1C2=CC3=C(C=C2)N=C(N3)C=CC4=CC=C(C=C4)C(F)(F)F)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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