MK-1421

Catalog No.: A63912
sstr3 Antagonist
MK-1421 is a potent and selective antagonist of the somatostatin receptor type 3 (sstr3). By inhibiting sstr3, MK-1421 plays a significant role in the modulation of insulin secretion, making it a valuable tool in research related to type 2 diabetes. Its specificity and efficacy make it suitable for investigating the complex pathways involved in metabolic disorders.
Grouped product items
Size Price Stock Qty
25mg
$1,530.00
In stock
50mg
$1,950.00
In stock
100mg
$2,480.00
In stock
Bulk Size
Bulk Discount
Free Delivery on orders over $500
Research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
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Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
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Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionMK-1421 is a potent and selective antagonist of the somatostatin receptor type 3 (sstr3). By inhibiting sstr3, MK-1421 plays a significant role in the modulation of insulin secretion, making it a valuable tool in research related to type 2 diabetes. Its specificity and efficacy make it suitable for investigating the complex pathways involved in metabolic disorders.
Product Information
Catalog NumA63912
FormulaC27H24FN9O2
Molecular Weight525.54
CAS Number1235995-16-0
SMILESFC(C=C1)=CN=C1C2=CNC([C@@H]3N[C@@](C4=CN(CC)N=C4)(C5=NN(C)C(O5)=O)C6=C(C(C=CC=C7)=C7N6)C3)=N2
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