MK-4256

Catalog No.: A21510

SSTR3 antagonist

MK-4256

MK-4256 Chemical Structure

CAS NO. 1104599-69-0

MK-4256 is a potent and selective SSTR3 antagonist with IC50s of 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively.

Availability: In stock

Package Price Qty
1 mg
$162.00
5 mg
$486.00
10 mg
$828.00
50 mg
$2,484.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

MK-4256 is a potent and selective SSTR3 antagonist with IC50s of 0.66 nM and 0.36 nM in human and mouse receptor binding assays, respectively.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.22 mL 101.11 mL 202.22 mL
0.5 mM 4.04 mL 20.22 mL 40.44 mL
1 mM 2.02 mL 10.11 mL 20.22 mL
5 mM 0.4 mL 2.02 mL 4.04 mL

*The above data is based on the productmolecular weight 494.52. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21510
Actions Antagonist
CAS No. 1104599-69-0
Formula C27H23FN8O
M. Wt 494.52
Solubility DMSO
Purity >98%
Synonyms MK4256; MK 4256
SMILES CN1N=CC([[email protected]@]2(C3=NOC(C)=N3)N[[email protected]@H](C4=NC=C(C5=CC=C(F)C=C5)N4)CC6=C2NC7=C6C=CC=C7)=C1
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy MK-4256 | MK-4256 Supplier | purchase | cost | manufacturer | order | distributor | buy 1104599-69-0| 1104599-69-0 Supplier | purchase 1104599-69-0 | 1104599-69-0 cost | 1104599-69-0 manufacturer | order 1104599-69-0 | 1104599-69-0 distributor
Rewards