Mozavaptan-d6 is a deuterium-labeled variant of Mozavaptan, a selective competitive antagonist of the vasopressin V2 receptor, with an IC50 of 14 nM. This compound exhibits approximately 85-fold selectivity for the V2 receptor compared to the V1 receptor, which has an IC50 of 1.2 μM. Mozavaptan-d6 is utilized in research studying the modulation of fluid balance and potential therapies for hyponatremia, syndrome of inappropriate antidiuretic hormone secretion (SIADH), and congestive heart failure. Its stable isotope labeling enables advanced pharmacokinetic studies and metabolic profiling.
Mozavaptan-d6 is a deuterium-labeled variant of Mozavaptan, a selective competitive antagonist of the vasopressin V2 receptor, with an IC50 of 14 nM. This compound exhibits approximately 85-fold selectivity for the V2 receptor compared to the V1 receptor, which has an IC50 of 1.2 μM. Mozavaptan-d6 is utilized in research studying the modulation of fluid balance and potential therapies for hyponatremia, syndrome of inappropriate antidiuretic hormone secretion (SIADH), and congestive heart failure. Its stable isotope labeling enables advanced pharmacokinetic studies and metabolic profiling.
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