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MRS4596

Catalog No.: A67917
P2X4 Receptor Antagonist
MRS4596 is a potent and selective antagonist of the P2X4 receptor, exhibiting an IC50 value of 1.38 μM for the human P2X4 receptor. This compound demonstrates neuroprotective and neuro-rehabilitative effects in models of ischemic stroke. MRS4596 is applicable in the study of ischemic stroke and associated therapeutic strategies.
MRS4596 2840581-38-4 P2X4 Receptor Antagonist
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Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionMRS4596 is a potent and selective antagonist of the P2X4 receptor, exhibiting an IC50 value of 1.38 μM for the human P2X4 receptor. This compound demonstrates neuroprotective and neuro-rehabilitative effects in models of ischemic stroke. MRS4596 is applicable in the study of ischemic stroke and associated therapeutic strategies.
Product Information
Catalog NumA67917
FormulaC22H15N4NaO3S
Molecular Weight438.43
CAS Number2840581-38-4
SMILESO=C(C1)NC(C2=CC=C(C=C2C=C3)C)=C3N(C4=CC=CC(C([N-]5)=NOC5=S)=C4)C1=O.[Na+]
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Neuronal Signaling > P2X Receptor