Catalog No.: A19426

BRD3/4 degrader


MZP-54 Chemical Structure

CAS NO. 2010159-47-2

MZP-54 is a selective degrader of BRD3/4 based on PROTAC technology, with a Kd of 4 nM for Brd4BD2.

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Biological Activity

MZP-54 is a selective degrader of BRD3/4 based on PROTAC technology, with a Kd of 4 nM for Brd4BD2.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 9.65 mL 48.23 mL 96.46 mL
0.5 mM 1.93 mL 9.65 mL 19.29 mL
1 mM 0.96 mL 4.82 mL 9.65 mL
5 mM 0.19 mL 0.96 mL 1.93 mL

*The above data is based on the productmolecular weight 1036.67. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A19426
Actions Degrader
CAS No. 2010159-47-2
Formula C55H66ClN7O9S
M. Wt 1036.67
Purity >98%
Synonyms MZP54, MZP 54
SMILES O=C(NCCOCCOCCOCC(N[[email protected]@H](C(C)(C)C)C(N1C[[email protected]](O)C[[email protected]]1C(NCC2=CC=C(C3=C(C)N=CS3)C=C2)=O)=O)=O)C(C=C4)=CC=C4C5=CC6=C(C=C5)N(C(C)=O)[[email protected]@H](C)C[[email protected]]6NC7=CC=C(Cl)C=C7

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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