N-Desethyl Sunitinib

Catalog No.: A15182

VEGFR/PDGFRβ/KIT inhibitor

N-Desethyl Sunitinib Chemical Structure

CAS NO. 356068-97-8

N-desethyl sunitinib is a major and pharmacologically active metabolite of sunitinib, which is potent, ATP-competitive VEGFR, PDGFRβ and KIT inhibitor (Ki values are 2, 9, 17, 8 and 4 nM for VEGFR -1, -2, -3, PDGFRβ and KIT respectively).

Availability: In stock

Package Price Qty
5 mg
$225.00
10 mg
$315.00
50 mg
$785.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

N-desethyl sunitinib is a major and pharmacologically active metabolite of sunitinib, which is potent, ATP-competitive VEGFR, PDGFRβ and KIT inhibitor (Ki values are 2, 9, 17, 8 and 4 nM for VEGFR -1, -2, -3, PDGFRβ and KIT respectively).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 27 mL 134.98 mL 269.96 mL
0.5 mM 5.4 mL 27 mL 53.99 mL
1 mM 2.7 mL 13.5 mL 27 mL
5 mM 0.54 mL 2.7 mL 5.4 mL

*The above data is based on the productmolecular weight 370.42. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A15182
Actions Inhibitor
M. Wt 370.42
Formula C20H23FN4O2
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 356068-97-8
Synonyms SU11662, SU 11662, SU-11662
SMILES CCNCCNC(=O)C1=C(NC(=C1C)C=C2C3=C(C=CC(=C3)F)NC2=O)C

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