Total item
Cart Subtotal
$0.00 Customer Appreciation Sale.
15% off with promo code "APPRECIATION2023" on check out or purchase order
Biological Activity
Nazartinib mesylate (EGF816 mesylate) is a novel, covalent mutant-selective EGFR inhibitor, with Ki and Kinact of 31 nM and 0.222 min?1 on EGFR(L858R/790M) mutant, respectively.
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 16.92 mL | 84.59 mL | 169.17 mL |
| 0.5 mM | 3.38 mL | 16.92 mL | 33.83 mL |
| 1 mM | 1.69 mL | 8.46 mL | 16.92 mL |
| 5 mM | 0.34 mL | 1.69 mL | 3.38 mL |
*The above data is based on the productmolecular weight 591.12. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A21741 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 1508250-72-3 |
| Formula | C27H35ClN6O5S |
| M. Wt | 591.12 |
| Purity | >98% |
| Synonyms | EGF816 (mesylate), EGF 816, EGF-816 |
| SMILES | O=C(C1=CC(C)=NC=C1)NC2=NC3=CC=CC(Cl)=C3N2[C@H]4CN(C(/C=C/CN(C)C)=O)CCCC4.CS(=O)(O)=O |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
Product Tags
Product Questions
Product Questions
No Questions
Keywords:buy Nazartinib mesylate | Nazartinib mesylate Supplier | purchase | cost | manufacturer | order | distributor | buy 1508250-72-3| 1508250-72-3 Supplier | purchase 1508250-72-3 | 1508250-72-3 cost | 1508250-72-3 manufacturer | order 1508250-72-3 | 1508250-72-3 distributor
Adooq Quality Guarantee
We promise all products perform as described.