NVP-BAG956

Catalog No.: A11511

PI3K/PDK-1 Inhibitor

NVP-BAG956

NVP-BAG956 Chemical Structure

CAS NO. 853910-02-8

NVP-BAG956 acts as a potent, reversible, and ATP-competitive PI 3-K/PDK1 dual kinase inhibitor, displaying much reduced potency against VEGFR1 (IC50 = 2.56 uM) and little or no activity toward a panel of 15 other kinases (IC50 >10 uM).

Availability: In stock

Package Price Qty
5 mg
$80.00
10 mg
$140.00
25 mg
$280.00
50 mg
$480.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

NVP-BAG956 acts as a potent, reversible, and ATP-competitive PI 3-K/PDK1 dual kinase inhibitor, displaying much reduced potency against VEGFR1 (IC50 = 2.56 uM) and little or no activity toward a panel of 15 other kinases (IC50 >10 uM).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.39 mL 116.96 mL 233.92 mL
0.5 mM 4.68 mL 23.39 mL 46.78 mL
1 mM 2.34 mL 11.7 mL 23.39 mL
5 mM 0.47 mL 2.34 mL 4.68 mL

*The above data is based on the productmolecular weight 427.5 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11511
Actions Inhibitor
M. Wt 427.5
Formula C28H21N5
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 853910-02-8
Synonyms NVP-BAG 956
SMILES CC1=NC2=CN=C3C=CC(=CC3=C2N1C4=CC=C(C=C4)C(C)(C)C#N)C#CC5=CN=CC=C5

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