Catalog No.
Product Name
Application
Product Information
Citations
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Drug Derivative
Haptamide B is a novel drug derivative with demonstrated biological activity. This compound primarily functions as an active ingredient in pharmacological applications, exhibiting potential in various therapeutic domains. Its unique structure and mechanism of action make it a valuable tool for research pertaining to drug development and optimization. -
Drug Derivative
8-iso Prostaglandin F1α is a prostaglandin derivative that exhibits potent biological activity by modulating various receptor pathways. It has been shown to play a role in inflammatory responses and may affect vascular function. This compound is utilized in research applications involving cardiovascular biology and inflammation studies, providing insights into the physiological effects of prostaglandins in disease models. -
Drug Derivative
Lopirazepam is a benzodiazepine derivative that primarily acts as a positive allosteric modulator of GABA-A receptors. It exhibits anxiolytic and sedative properties, making it valuable for research into anxiety disorders and sleep regulation. This compound is useful for studying the pharmacological effects of benzodiazepines and their potential therapeutic applications in neuropharmacology. -
Drug Derivative
Ascrolimus is a drug derivative that acts primarily as an immunosuppressant by inhibiting the mechanistic target of rapamycin (mTOR). This compound demonstrates significant biological activity in modulating immune responses, making it valuable for research in transplantation and autoimmune disease therapies. Its application extends to studying cell proliferation, growth regulation, and the underlying mechanisms of various diseases linked to mTOR signaling pathways. -
Drug Derivative
3,4-Methylenedioxy PV8 hydrochloride is a synthetic drug derivative featuring a pyrrolidine structure. This compound exhibits biological activity relevant for pharmacological research, particularly in studies aimed at understanding its effects on neurotransmitter systems. It serves as a valuable tool for investigating the mechanisms of action of related compounds and contributes to the development of novel therapeutic agents. -
Drug Derivative
N-Methoxy mephedrone hydrochloride is a derivative of mephedrone, primarily targeting monoamine transporters. This compound exhibits stimulant properties and can influence serotonin and dopamine release, making it valuable for research in neuropharmacology. Its applications extend to studies investigating psychostimulant effects and the development of new therapeutic strategies for mood disorders. -
Drug Derivative
CEP-2563 is a selective drug derivative with a focus on modulating key signaling pathways. It has demonstrated potential in various biological assays, particularly in the context of cancer research and cellular signaling investigations. Further studies can explore its efficacy and mechanism of action in targeted therapies and novel drug development. -
Drug Derivative
Styramate is a drug derivative that exhibits significant biological activity by modulating key biological pathways. It has been explored for its potential therapeutic applications in various disease models, contributing to research in pharmacology and drug development. Studies on Styramate can aid in understanding its mechanism of action and efficacy in targeted treatments. -
Drug Derivative
ML67 is a potent drug derivative that inhibits specific biological pathways. This compound exhibits significant activity in modulating cellular processes, making it valuable for research in pharmacology and drug development. Its application extends to studying the mechanisms of action of related therapeutics and exploring novel therapeutic strategies. -
Drug Derivative
N-Methyl benzedrone hydrochloride is a drug derivative primarily known for its stimulant properties. It acts as a monoamine reuptake inhibitor, enhancing the levels of neurotransmitters such as dopamine and norepinephrine in the brain. This compound is utilized in research focused on neuropharmacology, studying its effects on mood, cognition, and potential therapeutic applications. Its relevance in the analysis of psychostimulant behaviors and drug interactions makes it a valuable reagent in chemical research. -
Drug Derivative
Triethylene glycol diacetate is an orally active derivative of triethylene glycol that targets reproductive toxicity pathways. This compound has been demonstrated to reduce body weights in nursing mouse pups during lactation, with effects that reverse by young adulthood. Additionally, it increases the combined kidney and adrenal weight in adult specimens. Triethylene glycol diacetate is valuable for investigating reproductive and developmental toxicity in preclinical research. -
Drug Derivative
AZD6370 is a selective drug derivative that targets the protein kinase PI3K. This compound exhibits potent inhibition of PI3K activity, making it a valuable tool for studying cellular signaling pathways and metabolic regulation. It is utilized in research focused on cancer biology, specifically in evaluating therapeutic strategies that disrupt PI3K-mediated signaling. -
Drug Derivative
Prodiamine is a potent drug derivative known for its selective inhibition of certain biological pathways. It displays significant anti-inflammatory properties, making it suitable for research applications in pharmacology and toxicology. Prodiamine is often utilized in studies investigating drug metabolism and efficacy, contributing valuable insights into the development of therapeutic agents. -
Drug Derivative
Mesulergine is a drug derivative that primarily targets serotonin receptors. This compound exhibits notable effects on neurotransmission, making it relevant in studies related to neuropharmacology and psychiatric disorders. Its potential applications include investigating the mechanisms of psychotropic effects and exploring therapeutic avenues for mood regulation and anxiety disorders. -
Drug Derivative
Amicarbalide is a drug derivative known for its inhibitory effects on monoamine oxidase (MAO). This compound exhibits biological activity by modulating neurotransmitter levels, making it useful in research related to neurodegenerative diseases and mood disorders. Its ability to influence monoamine metabolism renders it a valuable tool in the study of pharmacological mechanisms underlying depression and anxiety. -
Drug Derivative
Dihydro-β-ionol is a derivative of β-Ionone, primarily targeting intracellular melanin synthesis. This compound has demonstrated significant inhibitory effects on melanin production, making it a valuable tool in cancer research, particularly in the study of melanoma. Its unique properties facilitate investigations into mechanisms of pigmentation and potential therapeutic strategies in skin cancers. -
Drug Derivative
AP23846 is a drug derivative known for its modulation of cellular pathways involved in various biological processes. It exhibits significant bioactivity that can be utilized in pharmacological profiling and research applications focused on drug discovery and development. This compound serves as a valuable tool for investigating therapeutic effects and mechanisms of action in targeted treatments. -
Drug Derivative
Etoposide toniribate is a derivative of etoposide, primarily acting as a topoisomerase II inhibitor. It exhibits cytotoxic activity against a wide range of cancer cell lines, making it a valuable tool in cancer research. This compound is utilized in studies focused on elucidating mechanisms of drug resistance and evaluating therapeutic efficacy in various oncological settings. -
Drug Derivative
Isocil is a drug derivative that exhibits notable pharmacological activity. It has been investigated for its potential effects on various biological pathways, making it a valuable tool in drug development research. Its applications extend to studying drug metabolism and interactions in cellular models, contributing to the understanding of therapeutic efficacy and safety profiles. -
Drug Derivative
42-O-(2-Aminoethyl)-rapamycin is a derivative of the mTOR inhibitor rapamycin, targeting the mechanistic target of rapamycin (mTOR) pathway. This compound exhibits potential for pharmaceutical research, particularly in the development of conjugates, by enhancing the bioactivity of rapamycin while maintaining its functional properties. Its application in drug development can facilitate advancements in therapeutic strategies against various diseases, including cancer and metabolic disorders. -
Drug Derivative
Muraglitazar glucuronide is a glucuronide derivative of the drug Muraglitazar, primarily targeting peroxisome proliferator-activated receptors (PPARs). This compound exhibits potent agonistic activity towards PPARα and PPARγ, playing a significant role in lipid metabolism and glucose homeostasis. Research applications include studying metabolic disorders, diabetes, and cardiovascular diseases, providing insights into the pharmacological effects of PPAR modulation. -
Drug Derivative
Darcanolide is a drug derivative known for its potential pharmacological activity. It exhibits notable effects in various biological systems, making it a valuable tool in chemical research and drug development. Its applications include the investigation of drug interactions and the modulation of biological pathways. As a compound of interest, Darcanolide contributes to advancing our understanding of medicinal chemistry and therapeutic strategies. -
Drug Derivative
Ambasilide is a drug derivative with known efficacy in modifying biological responses. It exhibits significant activity in cellular pathways related to inflammation and cell proliferation. This compound is primarily utilized in research focused on drug development and therapeutic applications. -
Drug Derivative
OX3a is a potent drug derivative with demonstrated biological activity. This compound is primarily utilized in research focused on drug development and mechanism of action studies. Its unique properties make it suitable for exploring therapeutic interventions and understanding drug-receptor interactions in various biological systems. -
Drug Derivative
4-Methyl-α-pyrrolidinoisohexanophenone hydrochloride is a drug derivative that primarily targets the monoamine transporter system. It exhibits stimulant and psychoactive properties, making it a valuable tool in neuropharmacological research. This compound may be utilized in studies investigating the mechanisms of drug action and the effects of novel psychoactive substances on neurotransmitter dynamics. -
Drug Derivative
7-Descarbamoyl-17-amino geldanamycin is a derivative of Geldanamycin, targeting the heat shock protein 90 (HSP90). This compound demonstrates limited activity in the degradation of the p185erbB-2 protein within human breast cancer cells in vitro. It serves as a useful tool for investigating the role of HSP90 inhibition in cancer biology and can aid in the development of therapeutic strategies against breast cancer. -
Drug Derivative
3',4'-Dimethyl-α-ethylaminovalerophenone hydrochloride is a synthetic drug derivative known for its psychoactive properties. It primarily functions as a selective monoamine reuptake inhibitor, influencing neurotransmitter levels in the central nervous system. This compound is utilized in research related to neuropharmacology and drug development, particularly in the study of substance abuse and therapeutic applications. -
Drug Derivative
N-Propyl hexylone hydrochloride is a synthetic derivative targeting various neurochemical pathways. This compound is primarily studied for its stimulant properties and potential effects on the monoamine system, particularly concerning dopamine and norepinephrine reuptake inhibition. Its applications include research into psychoactive substances, behavioral studies, and investigations of drug addiction. -
Drug Derivative
[Gly9-OH]-Atosiban is a derivative of Atosiban, primarily targeting the oxytocin receptor. This compound exhibits antagonistic activity, making it valuable for research focused on uterine contractions and labor modulation. It is particularly useful in studies investigating the physiological effects of oxytocin in reproductive health and related disorders. -
Drug Derivative
(Z)-8-Dodecenyl acetate is a drug derivative known for its role as a pheromone and chemical signaling molecule. It exhibits biological activity related to insect attraction and communication, making it valuable for research in entomology and pest management. This compound can be employed in studies focused on behavioral responses in insects, offering insights into ecological interactions and potential applications in biocontrol strategies. -
Drug Derivative
3-Isomangostin hydrate formate is a derivative of the natural product mangostin, isolated from the fruit of Garcinia mangostana Linn. This compound exhibits significant biological activity and has been studied for its potential therapeutic effects, particularly in the fields of anti-inflammatory research and cancer treatment. Its unique structure and properties make it a valuable reagent for various biological assays and investigations into the pharmacological potential of mangosteen components. -
Drug Derivative
14,15-Leukotriene A4 methyl ester is a methyl ester derivative of Leukotriene A4, primarily utilized to investigate the biological effects of leukotrienes. This compound plays a significant role in inflammation and immune response, making it a valuable tool for research in pharmacology and biochemistry. Its ability to modulate leukotriene pathways allows for in-depth studies related to various inflammatory conditions and potential therapeutic targets. -
Drug Derivative
Lab 170250F is a drug derivative known for its potent biological activity. It serves as an essential reagent for drug discovery and development, particularly in the synthesis and evaluation of pharmacological properties. This compound facilitates the exploration of therapeutic mechanisms and aids in the design of novel drug candidates. Its application spans various fields, including medicinal chemistry and pharmacology research. -
Drug Derivative
L 365031 is a potent drug derivative that targets specific receptors involved in cellular signaling pathways. This compound exhibits significant biological activity, making it a valuable tool for research applications in pharmacology and drug development studies. Investigations utilizing L 365031 can enhance understanding of receptor-ligand interactions and contribute to the design of novel therapeutic agents. -
Drug Derivative
SU-13197 is a potent drug derivative known for its inhibitory effects targeting specific molecular pathways. This compound exhibits significant biological activity, making it a valuable tool in research aimed at exploring therapeutic options for various diseases. Its applications extend to studies in pharmacology and drug development, providing insights into compound behavior and potential efficacy. -
Drug Derivative
JNJ-28330835 is a potent drug derivative primarily targeting specific cell signaling pathways. This compound has been shown to exhibit significant biological activity, making it valuable in the study of disease mechanisms and therapeutic interventions. Its applications extend to various fields of biomedical research, including cancer studies and pharmacological investigations. -
Heroin Impurity
ATM4 4-Acetoxy analog is identified as an impurity associated with the synthesis of heroin. This compound plays a notable role in chemical research related to opioid synthesis and quality control. Its characterization is crucial for understanding the intricacies of heroin production and ensuring regulatory compliance within drug development processes. -
Drug Derivative
GW813893 is a synthetic derivative designed to interact with specific molecular targets involved in cellular signaling pathways. This compound exhibits notable biological activity, making it useful for exploring mechanisms of action in pharmacological research. Its applications include investigating potential therapeutic effects and understanding drug-receptor interactions in disease models. -
Drug Derivative
GR 100679 is a drug derivative that acts as a selective antagonist. This compound exhibits significant biological activity in modulating receptor interactions, making it valuable for research in pharmacology and drug discovery. Its applications may include studying receptor signaling pathways and assessing therapeutic potential in various disease models. -
Drug Derivative
Sunitinib carboxylic acid is a carboxylic acid metabolite of Sunitinib, a multi-target tyrosine kinase inhibitor. This compound primarily targets receptor tyrosine kinases involved in angiogenesis and tumor growth, making it relevant for research on malignant tumors, including gastrointestinal stromal tumors, renal cell carcinoma, and pancreatic neuroendocrine tumors. Its role as a drug derivative provides insights into pharmacokinetics and efficacy in cancer therapy. -
Drug Derivative
SB209995 is a selective drug derivative that acts as a potent inhibitor of the protein kinase C (PKC) pathway. It exhibits significant biological activity by modulating cellular signaling processes associated with cell growth and differentiation. This compound is primarily utilized in research applications investigating cancer biology and therapeutic strategies aimed at PKC-related signaling pathways. -
Drug Derivative
Luminespib analog is a potent derivative targeting heat shock protein 90 (HSP90). It exhibits significant inhibitory activity, disrupting cancer cell proliferation and promoting apoptosis. This compound is valuable in cancer research, particularly in studies aimed at understanding the role of HSP90 in tumorigenesis and therapeutic resistance. -
Drug Derivative
Drazoxolon, a drug derivative, exhibits significant biological activity through its modulation of specific biochemical pathways. It is primarily utilized in research applications focused on investigating therapeutic potential in various disease models. This compound serves as a valuable tool in the exploration of pharmaceutical development and the understanding of drug action mechanisms. -
Drug Derivative
BVdUMP is a nucleotide analog that acts as a potent inhibitor of DNA synthesis. It exhibits significant biological activity by inhibiting the enzyme DNA polymerase and integrating into the DNA strand, leading to the disruption of nucleic acid metabolism. BVdUMP is primarily utilized in cancer research and studies focused on antiviral therapies, providing valuable insights into cellular proliferation and viral replication mechanisms. -
Drug Derivative
γ-Secretase modulator 16 is a selective modulator of the γ-secretase complex, primarily targeting the processing of amyloid precursor protein (APP). This compound is known to influence the production of amyloid-beta peptides, thereby playing a crucial role in the modulation of neurodegenerative pathways associated with Alzheimer's disease. It serves as a valuable tool for research aimed at understanding γ-secretase function and the development of therapeutic strategies for Alzheimer’s and other related disorders. -
Drug Derivative
BX048 is a potent drug derivative that acts as a selective modulator of target pathways. This compound exhibits significant biological activity, making it suitable for various research applications, including pharmacological studies and mechanism of action investigations. Researchers can utilize BX048 to explore its effects on cellular processes and therapeutic potential in specific disease models. -
Drug Derivative
A60586 is a synthetic derivative with a defined mechanism of action targeting specific biological pathways. It exhibits potent biological activity that makes it applicable for research in drug development and pharmacology. A60586 is particularly useful for studying the effects of drug modifications on efficacy and safety in various cellular and animal models. -
Drug Derivative
ACAT Inhibitor 1 is a potent inhibitor of acyl-CoA:cholesterol acyltransferase (ACAT), which is involved in cholesterol metabolism. This compound exhibits significant inhibitory activity in lipid accumulation and is useful in research related to atherosclerosis and metabolic disorders. It provides a valuable tool for investigating the role of ACAT in cellular lipid homeostasis and potential therapeutic strategies for cholesterol-related diseases. -
Drug Derivative
3,4-Methylenedioxy PV9 hydrochloride is a drug derivative that targets various cellular pathways associated with tumorigenesis. This compound exhibits cytotoxic effects on multiple human cancer cell lines, including BEAS-2B, aortic endothelial cells, HASM, SK-N-SH, A172, HepG2, MKN45, and DLD1, with lethal concentration (LC50) values ranging from 12.8 to 67.5 μM. Its biological activity supports research in cancer therapeutics and elucidation of mechanisms underlying cell death. -
Drug Derivative
ReN 1869 is a potent drug derivative that exhibits significant bioactivity through its interaction with specific molecular targets. This compound is primarily utilized in pharmacological research to explore its effects on cellular mechanisms and potential therapeutic applications. Its unique profile makes it a valuable tool in the investigation of drug development and efficacy studies.
