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Panulisib (P7170, AK151761)

Catalog No.: A14379

PI3K inhibitor

Panulisib (P7170, AK151761)

Panulisib (P7170, AK151761) Chemical Structure

CAS NO. 1356033-60-7

Panulisib is a potent and selective imidazoquinoline based PI3K inhibitor with potential anticancer activity.

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5 mg
$350.00
10 mg
$600.00
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Biological Activity

Biological Activity

Panulisib is a potent and selective imidazoquinoline based PI3K inhibitor with potential anticancer activity.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.96 mL 94.79 mL 189.57 mL
0.5 mM 3.79 mL 18.96 mL 37.91 mL
1 mM 1.9 mL 9.48 mL 18.96 mL
5 mM 0.38 mL 1.9 mL 3.79 mL

*The above data is based on the productmolecular weight 527.50321. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A14379
Actions Inhibitor
CAS No. 1356033-60-7
Formula C27H20F3N9
M. Wt 527.50321
Purity >98%
Synonyms AK151761, AK 151761, AK-151761
SMILES CC(C)(C#N)C1=NC=C(C=C1)N2C3=C4C=C(C=CC4=NC=C3N(C2=NC#N)C)C5=CC(=C(N=C5)N)C(F)(F)F
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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