PAT-1251 Hydrochloride

Catalog No.: A21969

LOXL2 inhibitor

PAT-1251 Hydrochloride

PAT-1251 Hydrochloride Chemical Structure

CAS NO. 2098884-53-6

PAT-1251 Hydrochloride is a potent, selective and oral lysyl oxidase-like 2 (LOXL2) inhibitor, with IC50s of 0.71 and 1.17 μM for hLOXL2 and hLOXL3, respectively, and also potently inhibits mouse, rat, and dog LOXL2 (IC50s, 0.10, 0.12, and 0.16 μM, respectively).

Availability: In stock

Package Price Qty
1 mg
$320.00
5 mg
$960.00
10 mg
$1,600.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

PAT-1251 Hydrochloride is a potent, selective and oral lysyl oxidase-like 2 (LOXL2) inhibitor, with IC50s of 0.71 and 1.17 μM for hLOXL2 and hLOXL3, respectively, and also potently inhibits mouse, rat, and dog LOXL2 (IC50s, 0.10, 0.12, and 0.16 μM, respectively).
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.95 mL 114.73 mL 229.46 mL
0.5 mM 4.59 mL 22.95 mL 45.89 mL
1 mM 2.29 mL 11.47 mL 22.95 mL
5 mM 0.46 mL 2.29 mL 4.59 mL

*The above data is based on the productmolecular weight 435.8. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21969
Actions Inhibitor
M. Wt 435.8
Formula C18H18ClF4N3O3
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 2098884-53-6
Synonyms PAT 1251, PAT1251
SMILES O=C(C1=CC=CC(OC2=NC(C(F)(F)F)=CC(CN)=C2)=C1)N3C[[email protected]@H](F)[[email protected]](O)C3.Cl

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