Trusted by 10,000+ Scientists since 2006



PAK4 inhibitor

0 Customer Reviews
Catalog No. A11930

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
PF-3758309 5mg A11930-5

Regular Price: $50.00

Special Price: $45.00

PF-3758309 10mg A11930-10

Regular Price: $80.00

Special Price: $72.00

PF-3758309 25mg A11930-25

Regular Price: $150.00

Special Price: $135.00

PF-3758309 50mg A11930-50

Regular Price: $240.00

Special Price: $216.00

Adooq中国网址: www.adooq.cn全国免费电话: 400-025-6535 [email protected]

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

PF-3758309 is a small-molecule p21-activated kinase inhibitor inhibiting oncogenic signaling and tumor growth.


Double click on above image to view full picture

Zoom Out
Zoom In

More Views

Publications citing Adooq Products

Chemical Information

Catalog Num A11930
Actions Inhibitor
M. Wt 490.2
Formula C25H30N8OS
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 898044-15-0
Synonyms PF-03758309
SMILES CC1=NC2=C(C(=N1)NC3=NNC4=C3CN(C4(C)C)C(=O)N[[email protected]](CN(C)C)C5=CC=CC=C5)SC=C2

Biological Activity

PF-3758309 is a small-molecule p21-activated kinase inhibitor inhibiting oncogenic signaling and tumor growth.
Target Value
PAK4IC50: 1.3nM
PAK1ki: 13.7nM
PAK6ki: 17.1nM
PAK5ki: 18.1nM
PAK4ki: 18.7nM
PAK3IC50: 99nM
PAK2IC50: 190nM

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.4 mL 102 mL 204mL
0.5 mM 4.08 mL 20.4 mL 40.8 mL
1 mM 2.04 mL 10.2 mL 20.4 mL
5 mM 0.41 mL 2.04 mL 4.08 mL

*The above data is based on the productmolecular weight 490.2 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

View Related Products By Research Topics

Cat. No.

Product NameSolubility(mg/mL)
A10255 ABT-737 <1 mg/mL 163 mg/mL <1 mg/mL
A10022 ABT-263 (Navitoclax) <1 mg/mL 195 mg/mL <1 mg/mL
A10665 Obatoclax mesylate (GX15-070) <1 mg/mL 83 mg/mL <1 mg/mL
A10955 TW-37 <1 mg/mL 115 mg/mL 4 mg/mL
A10984 VX-765 <1 mg/mL 102 mg/mL 102 mg/mL
A11090 PAC-1 <1 mg/mL 78 mg/mL 16 mg/mL
A10491 JNJ 26854165 <1 mg/mL 66 mg/mL 2 mg/mL
A11931 RITA (NSC 652287) <1 mg/mL 115 mg/mL 4 mg/mL
A10522 Lenalidomide (CC-5013) <1 mg/mL 52 mg/mL <1 mg/mL
A10743 Pomalidomide (CC-4047) <1 mg/mL 55 mg/mL <1 mg/mL
A11163 AT-406 <1 mg/mL 112 mg/mL 112 mg/mL
A11002 YM155 89 mg/mL 55 mg/mL 6 mg/mL
A10935 Tipifarnib (Zarnestra) <1 mg/mL 83 mg/mL <1 mg/mL
A10657 Nutlin-3 <1 mg/mL 116 mg/mL 116 mg/mL

Ordering online

To place an order online, simply browse to the product you are interested in and click on the 'Add to Cart' button. To complete this process, you will need to confirm the size and quantity of the products that you require.

To complete an order you will need to register using our simple online registration process. We do not share your contact details with any third parties.

When you are ready to check out simply enter your PO number to complete the ordering process. Please ensure that you send us a copy of your PO by fax or email afterwards.  We will then liaise with you or your purchasing department to confirm the order.

Found your products but not ready to order?

Why not use our WishList feature to store lists of products? This convenient feature allows you to manage lists, append notes to products and share lists with co-workers or colleagues.

Ordering offline

You can email or fax us your purchase order and we will place the order for you. You can also phone us to place the order.  Our contact details are:

We require the following information to process your order:
  • The catalog number for each product. 
  • Your email address or fax number. 
  • Your name and telephone number. 
  • Shipping address and billing address.
  • Purchase order numbers.

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Similar product(s)

Keywords:buy PF-3758309 | PF-3758309 Supplier | purchase PF-3758309 | PF-3758309 cost | PF-3758309 manufacturer | order PF-3758309 | PF-3758309 distributor | buy 898044-15-0| 898044-15-0 Supplier | purchase 898044-15-0 | 898044-15-0 cost | 898044-15-0 manufacturer | order 898044-15-0 | 898044-15-0 distributor