PF-3758309

Catalog No.: A11930

PAK4 inhibitor

PF-3758309 Chemical Structure

CAS NO. 898044-15-0

PF-3758309 is a small-molecule p21-activated kinase inhibitor inhibiting oncogenic signaling and tumor growth.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $50.00

Special Price $40.00

10 mg

Regular Price: $80.00

Special Price $64.00

25 mg

Regular Price: $150.00

Special Price $120.00

50 mg

Regular Price: $240.00

Special Price $192.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

PF-3758309 is a small-molecule p21-activated kinase inhibitor inhibiting oncogenic signaling and tumor growth.
Targets
Target Value
PAK4IC50: 1.3nM
PAK1ki: 13.7nM
PAK6ki: 17.1nM
PAK5ki: 18.1nM
PAK4ki: 18.7nM
PAK3IC50: 99nM
PAK2IC50: 190nM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 20.4 mL 102 mL 204 mL
0.5 mM 4.08 mL 20.4 mL 40.8 mL
1 mM 2.04 mL 10.2 mL 20.4 mL
5 mM 0.41 mL 2.04 mL 4.08 mL

*The above data is based on the productmolecular weight 490.2 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11930
Actions Inhibitor
M. Wt 490.2
Formula C25H30N8OS
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 898044-15-0
Synonyms PF-03758309
SMILES CC1=NC2=C(C(=N1)NC3=NNC4=C3CN(C4(C)C)C(=O)N[[email protected]](CN(C)C)C5=CC=CC=C5)SC=C2

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