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PKI-587 ( Gedatolisib )


PI3K/mTOR inhibitor

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Catalog No. A11079

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
PKI-587 5mg A11079-5

Regular Price: $50.00

Special Price: $45.00

PKI-587 10mg A11079-10

Regular Price: $90.00

Special Price: $81.00

PKI-587 50mg A11079-50

Regular Price: $360.00

Special Price: $324.00

PKI-587 100mg A11079-100

Regular Price: $680.00

Special Price: $612.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

PKI-587 is a highly potent PI3K/mTOR kinase inhibitor that inhibits PI3K-α,β,γ, δ isoforms and mTOR with IC50 of 0.4, 6.0, 5.4, 6.0 and 1.6 nM respectively.

PKI-587 ( Gedatolisib )

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Chemical Information

Catalog Num A11079
Actions Inhibitor
M. Wt 615.7
Formula C32H41N9O4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1197160-78-3
Synonyms PKI587, Gedatolisib

Biological Activity

PKI-587 is a highly potent PI3K/mTOR kinase inhibitor that inhibits PI3K-α,β,γ, δ isoforms and mTOR with IC50 of 0.4, 6.0, 5.4, 6.0 and 1.6 nM respectively.
PI3Kα (Cell-free assay) mTOR (Cell-free assay) PI3Kγ (Cell-free assay)
0.4 nM1.6 nM5.4 nM


Solubility (25°C)* In vitro DMSO 2 mg/mL (3.24 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 16.24 mL 81.21 mL 162.42mL
0.5 mM 3.25 mL 16.24 mL 32.48 mL
1 mM 1.62 mL 8.12 mL 16.24 mL
5 mM 0.32 mL 1.62 mL 3.25 mL

*The above data is based on the productmolecular weight 615.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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