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PRL 2915

Catalog No.: A63853
hsst2 Antagonist
PRL 2915 is a potent antagonist of the human somatostatin subtype 2 receptor (hsst2), exhibiting a Ki value of 12 nM. This compound effectively inhibits hsst2-mediated signaling pathways, making it a valuable tool for studying somatostatin-related physiological processes and disorders. Its application in research may contribute to a better understanding of neuroendocrine regulation and potential therapeutic approaches in related diseases.
PRL 2915 209006-18-8 hsst2 Antagonist
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Size Price Stock Qty
1mg
$25.00
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5mg
$50.00
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10mg
$85.00
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Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionPRL 2915 is a potent antagonist of the human somatostatin subtype 2 receptor (hsst2), exhibiting a Ki value of 12 nM. This compound effectively inhibits hsst2-mediated signaling pathways, making it a valuable tool for studying somatostatin-related physiological processes and disorders. Its application in research may contribute to a better understanding of neuroendocrine regulation and potential therapeutic approaches in related diseases.
Product Information
Catalog NumA63853
FormulaC59H71ClN12O8S2
Molecular Weight1175.85
CAS Number209006-18-8
Sequence{Phe<4-Cl>}-{d-Cys}-{β-Ala<3-Py>}-{d-Trp}-Lys-{Val<3-Me>}-Cys-{2-Nal}-NH2(Disulfide bond)
Sequence shortening{F<4-Cl>}-{d-C}-{β-A<3-Py>}-{d-W}-K-{V<3-Me>}-C-{A<3(2-Naph)>}-NH2 (Disulfide bridge:Cys2-Cys7)
SMILESCC(C)(C)[C@@H]1NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2cccnc2)NC(=O)[C@@H](CSSC[C@H](NC1=O)C(=O)N[C@@H](Cc1ccc2ccccc2c1)C(N)=O)NC(=O)[C@@H](N)Cc1ccc(Cl)cc1
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GPCR/G Protein > Somatostatin Receptors