R1530

Catalog No.: A13111

Chk2, KDR, FGFR, Aurora A & Cdk2 inhibitor

R1530

R1530 Chemical Structure

CAS NO. 882531-87-5

R1530 is a pyrazolobenzodiazepine small molecule with potential antiangiogenesis and antineoplastic activities. R1530 is also a mitosis-angiogenesis inhibitor (MAI) that inhibits multiple receptor tyrosine kinases involved in angiogenesis, such as vascular endothelial growth factor receptor (VEGFR)-1, -2, -3, platelet-derived growth factor receptor (PDGFR) beta? FMS-like tyrosine kinase (Flt)-3, and fibroblast growth factor receptor (FGFR) -1, -2.

Availability: In stock

Package Price Qty
5 mg
$60.00
10 mg
$100.00
25 mg
$200.00
50 mg
$320.00
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Warning WARNING: Attention California Residents: This product can expose you to chemicals including R1530 , which is known to the State of California to cause cancer and birth defects or other reproductive harm. For more information, go to www.P65Warnings.ca.gov
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

R1530 is a pyrazolobenzodiazepine small molecule with potential antiangiogenesis and antineoplastic activities. R1530 is also a mitosis-angiogenesis inhibitor (MAI) that inhibits multiple receptor tyrosine kinases involved in angiogenesis, such as vascular endothelial growth factor receptor (VEGFR)-1, -2, -3, platelet-derived growth factor receptor (PDGFR) beta? FMS-like tyrosine kinase (Flt)-3, and fibroblast growth factor receptor (FGFR) -1, -2.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 28.03 mL 140.14 mL 280.28 mL
0.5 mM 5.61 mL 28.03 mL 56.06 mL
1 mM 2.8 mL 14.01 mL 28.03 mL
5 mM 0.56 mL 2.8 mL 5.61 mL

*The above data is based on the productmolecular weight 356.78. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A13111
Actions Inhibitor
M. Wt 356.78
Formula C18H14ClFN4O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 882531-87-5
Synonyms R-1530, R 1530
SMILES CC1=C2C(=NC3=CC(=C(C=C3C(=N2)C4=CC=CC=C4Cl)F)OC)NN1

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