(Rac)-VU 6008667

Catalog No.: A21939

mAChR M5 negative allosteric modulator

(Rac)-VU 6008667

(Rac)-VU 6008667 Chemical Structure

CAS NO. 2092917-63-8

(Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM, pIC50= 5.75), has high CNS penetration.

Availability: In stock

Package Price Qty
5 mg
$162.00
10 mg
$279.00
50 mg
$828.00
100 mg
$1,656.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

(Rac)-VU 6008667 is a selective negative allosteric modulator of muscarinic acetylcholine receptor subtype 5 (M5 NAM) (IC50=1.8 μM, pIC50= 5.75), has high CNS penetration.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.79 mL 113.93 mL 227.87 mL
0.5 mM 4.56 mL 22.79 mL 45.57 mL
1 mM 2.28 mL 11.39 mL 22.79 mL
5 mM 0.46 mL 2.28 mL 4.56 mL

*The above data is based on the productmolecular weight 438.85. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A21939
Actions Modulator
CAS No. 2092917-63-8
Formula C24H17ClF2N2O2
M. Wt 438.85
Solubility DMSO
Purity >98%
Synonyms VU6008667, VU-6008667
SMILES O=C1N2C(N(C(C3=CC=C(F)C(F)=C3)=O)CC2)(C4=CC=C(Cl)C(C)=C4)C5=C1C=CC=C5
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Product Tags

Product Tags

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy (Rac)-VU 6008667 | (Rac)-VU 6008667 Supplier | purchase | cost | manufacturer | order | distributor | buy 2092917-63-8| 2092917-63-8 Supplier | purchase 2092917-63-8 | 2092917-63-8 cost | 2092917-63-8 manufacturer | order 2092917-63-8 | 2092917-63-8 distributor
Rewards