Biological Activity
Ralinepag is a potent, orally bioavailable and non-prostanoid prostacyclin (IP) receptor agonist, with EC50s of 8.5 nM, 530 nM and 850 nM for human and rat IP receptor and human DP1 receptor, respectively.
Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
---|---|---|---|
0.1 mM | 23.15 mL | 115.76 mL | 231.53 mL |
0.5 mM | 4.63 mL | 23.15 mL | 46.31 mL |
1 mM | 2.32 mL | 11.58 mL | 23.15 mL |
5 mM | 0.46 mL | 2.32 mL | 4.63 mL |
*The above data is based on the productmolecular weight 431.91. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
Catalog Num | A21073 |
---|---|
Actions | Agonist |
M. Wt | 431.91 |
Formula | C23H26ClNO5 |
Solubility | DMSO |
Purity | >98% |
Storage | at -20°C 3 years Powder |
CAS No. | 1187856-49-0 |
Synonyms | APD811, APD 811, APD-811 |
SMILES | O=C(O)COC[[email protected]]1CC[[email protected]](COC(N(C2=CC=C(Cl)C=C2)C3=CC=CC=C3)=O)CC1 |
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