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Rilmenidine-d4

Stable Isotope

Rilmenidine-d4 is a deuterium-labeled derivative of Rilmenidine, a selective I1 imidazoline receptor agonist and antihypertensive agent. It exhibits key biological activities including the induction of autophagy and modulation of apoptosis through the pro-apoptotic protein Bax in human leukemic K562 cells. Rilmenidine also operates centrally to reduce sympathetic overactivity and affects renal function by inhibiting the Na+/H+ antiport. This stable isotope is valuable for pharmacokinetic studies and mechanistic investigations in cardiovascular and cancer research.

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Specifications

Manufacturer	Adooq Bioscience
CAS Number	85047-14-9
Applications	Stable Isotope
Formula	C₁₀H₁₂D₄N₂O
Molecular Weight	184.27
SMILES	[2H]C1([2H])C([2H])(OC(NC(C2CC2)C3CC3)=N1)[2H]

Storage & Solubility

In Vitro Solubility

Reported Solubility

No reported solubility data are available for this product.

Preparing Stock Solutions

Stock preparation is unavailable for this product molecular weight.

Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.

Storage

Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.