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Publications citing Adooq Products
Chemical Information
| Catalog Num | A13272 |
|---|---|
| Actions | Inhibitor |
| M. Wt | 565.28 |
| Formula | C20H19F3IN3O5 |
| Solubility | DMSO |
| Purity | >98% |
| Storage | at -20°C 3 years Powder |
| CAS No. | 874101-00-5 |
| Synonyms | RO-4987655, RO 4987655 |
| SMILES | C1CC(=O)N(OC1)CC2=C(C(=C(C(=C2)C(=O)NOCCO)NC3=C(C=C(C=C3)I)F)F)F |
Description |
RO4987655 is an orally active small molecule, targeting mitogen-activated protein kinase kinase 1 (MAP2K1 or MEK1), with potential antineoplastic activity. | |||||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 17.69 mL | 88.45 mL | 176.9mL |
| 0.5 mM | 3.54 mL | 17.69 mL | 35.38 mL |
| 1 mM | 1.77 mL | 8.85 mL | 17.69 mL |
| 5 mM | 0.35 mL | 1.77 mL | 3.54 mL |
*The above data is based on the productmolecular weight 565.28. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
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