Catalog No.: A11143

TRPV1 antagonist


SB-705498 Chemical Structure

CAS NO. 501951-42-4

SB-705498 is a potent, selective and orally bioavailable TRPV1 antagonist.

Availability: In stock

Package Price Qty
5 mg
10 mg
50 mg
100 mg
10mM * 1mL in DMSO
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Biological Activity

SB-705498 is a potent, selective and orally bioavailable TRPV1 antagonist.
In vitro DMSO 78 mg/mL (181.71 mM)
Water Insoluble
Ethanol 18 mg/mL (41.93 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 23.36 mL 116.82 mL 233.64 mL
0.5 mM 4.67 mL 23.36 mL 46.73 mL
1 mM 2.34 mL 11.68 mL 23.36 mL
5 mM 0.47 mL 2.34 mL 4.67 mL

*The above data is based on the productmolecular weight 428.0 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A11143
Actions Antagonist
CAS No. 501951-42-4
Formula C17H16BrF3N4O
M. Wt 428.0
Purity >98%
Synonyms SB705498
SMILES C1CN(C[[email protected]@H]1NC(=O)NC2=CC=CC=C2Br)C3=NC=C(C=C3)C(F)(F)F

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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