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SST1 receptor antagonist-1

Catalog No.: A63911
SST1 Antagonist
SST1 receptor antagonist-1 is a selective antagonist of the Somatostatin receptor 1 (SST1), exhibiting pKds of 9.11 and 8.79 for rat and human SST1, respectively. This compound is utilized in research focused on retinal and endocrine dysfunctions, as well as cancer and neuropsychiatric disorders, making it a valuable tool for investigating the role of SST1 in various biological systems.
SST1 receptor antagonist-1 868057-23-2 SST1 Antagonist
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Research use only. We do not sell to patients.
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Adooq Products cited in reputable paper
Science VOLUME 380, ISSUE 6663 (2023)
Science VOLUME 369, ISSUE 6510 (2020)
Science VOLUME 356, ISSUE 6336 (2017)
Cell Vol. 185 Issue 23 p4428-4447.e28
Cell Vol 177, Issue 7, p1933-1947.e25
Cell Vol 156, Issue 5, p857-1114
Nature Volume 622 Issue 7982 (2023)
Nature volume 620, pages890-897 (2023)
Nature volume 610, pages540-546 (2022)
Nature volume 588, pages83-88 (2020)
Nature volume 574, pages268-272 (2019)
Nature volume 573, pages539-545 (2019)
Nature volume 567, pages118-122 (2019)
Nature volume 551, pages639-643 (2017)
Nature volume 551, pages247-250 (2017)
Nature volume 548, pages356-360 (2017)
Nature volume 545, pages187-192 (2017)
Biological Activity
DescriptionSST1 receptor antagonist-1 is a selective antagonist of the Somatostatin receptor 1 (SST1), exhibiting pKds of 9.11 and 8.79 for rat and human SST1, respectively. This compound is utilized in research focused on retinal and endocrine dysfunctions, as well as cancer and neuropsychiatric disorders, making it a valuable tool for investigating the role of SST1 in various biological systems.
Product Information
Catalog NumA63911
FormulaC29H31F2N3O2
Molecular Weight491.57
CAS Number868057-23-2
SMILESO=C(CCN(CCC1C2=C(OC3=C1C=CC=C3)C=CC=C2)C)N4CCN(CC4)C5=CC=C(C(F)=C5)F
Useful Calculator

This calculator helps you calculate mass of compound based on solution concentration, volume and molecular weight in a specific solution using the formula:

Mass (mg) = Concentration (mM) × Volume (mL) × Molecular Weight (g/mol)

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Please check COA/MSDS for correct molecular weight.

Calculate the dilution required to prepare a stock solution.
This equation is commonly abbreviated as: C1V1 = C2V2

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GPCR/G Protein > Somatostatin Receptors