TAK-875 (Fasiglifam)

Name: TAK-875 (Fasiglifam)
SKU: A11018
Price: 100 USD
Rating: 5 (3 reviews)

Catalog No.: A11018

GPR agonist

Adooq's TAK-875 (Fasiglifam) has been cited by 3 publications

TAK-875 is a potent, selective, and orally bioavailable GPR40 agonist.

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Grouped product items
Product Name	Price	Stock
TAK-875 5mg	$100.00	In stock
TAK-875 10mg	$150.00	In stock
TAK-875 50mg	$450.00	In stock
TAK-875 100mg	$720.00	In stock
*TAK-875 10mM 1mL in DMSO**	$110.00	In stock
Bulk Size	Bulk Discount

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Important Notice: For research use only. We do not sell to patients.

Data Sheet

SDS

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Adooq Products cited in reputable paper

Adooq's TAK-875 (Fasiglifam) has been cited by 3 publications

Ying Liu, .et al. , Nucleic Acids Res, 2018, Oct 12; 46(18): 9864-9874 PMID: 30219861

Deborah A. Goldspink, .et al. , Mol Metab, 2018, Jan; 7: 90-101 PMID: 29167062

Hodaka Yamada, .et al. , Sci Rep, 2016, 6: 25912 PMID: 27180622

Biological Activity

Discription	TAK-875 is a potent, selective, and orally bioavailable GPR40 agonist.

Product Information

Catalog Num	A11018
Formula	C29H32O7S
Molecular Weight	524.6
CAS Number	1000413-72-8
SMILES	CC1=C(C2=CC(COC3=CC=C([C@H](CC(O)=O)CO4)C4=C3)=CC=C2)C(C)=CC(OCCCS(C)(=O)=O)=C1
Synonyms	TAK875
Storage	Store lyophilized at -20ºC, keep desiccated. In lyophilized form, the chemical is stable for 36 months. In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

Solubility

In vitro (25°C)	DMSO	92 mg/mL (172.4 mM)
	Water	Insoluble
	Ethanol	Insoluble
In vivo	0.5% CMC+0.25% Tween 80	28 mg/mL
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass	1 mg	5 mg	10 mg
0.1 mM	19.06 mL	95.31 mL	190.62 mL
0.5 mM	3.81 mL	19.06 mL	38.12 mL
1 mM	1.91 mL	9.53 mL	19.06 mL
5 mM	0.38 mL	1.91 mL	3.81 mL

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