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TAK-875 (Fasiglifam)


GPR agonist

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Catalog No. A11018

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
TAK-875 5mg A11018-5

Regular Price: €95.00

Special Price: €85.50

TAK-875 10mg A11018-10

Regular Price: €142.50

Special Price: €128.25

TAK-875 50mg A11018-50

Regular Price: €427.50

Special Price: €384.75

TAK-875 100mg A11018-100

Regular Price: €684.00

Special Price: €615.60

TAK-875 10mM * 1mL in DMSO A11018-10mM-D

Regular Price: €104.50

Special Price: €94.05

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

TAK-875 is a potent, selective, and orally bioavailable GPR40 agonist.

TAK-875 (Fasiglifam)

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Publications citing Adooq Products
TAK-875 (Fasiglifam) Citations (3)
  • Ying Liu, .et al. A synthetic free fatty acid-regulated transgene switch in mammalian cells and mice, Nucleic Acids Res, 2018, Oct 12; 46(18): 9864-9874 PMID: 30219861
  • Deborah A. Goldspink, .et al. Mechanistic insights into the detection of free fatty and bile acids by ileal glucagon-like peptide-1 secreting cells, Mol Metab, 2018, Jan; 7: 90-101 PMID: 29167062
  • Hodaka Yamada, .et al. Potentiation of Glucose-stimulated Insulin Secretion by the GPR40-PLC-TRPC Pathway in Pancreatic β-Cells, Sci Rep, 2016, 6: 25912 PMID: 27180622

Chemical Information

Catalog Num A11018
Actions Agonist
M. Wt 533.6
Formula C29H32O7S.1/2H2O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1000413-72-8
Synonyms TAK875
SMILES CC1=CC(=CC(=C1C2=CC(=CC=C2)COC3=CC4=C(C=C3)[[email protected]@H](CO4)CC(=O)O)C)OCCCS(=O)(=O)C

Biological Activity

TAK-875 is a potent, selective, and orally bioavailable GPR40 agonist.


Solubility (25°C) * In vitro DMSO 100 mg/mL (187.39 mM)
Water <1 mg/mL (<1 mM)
Ethanol <1 mg/mL (<1 mM)
In vivo 0.5% CMC/0.25% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 18.74 mL 93.7 mL 187.41mL
0.5 mM 3.75 mL 18.74 mL 37.48 mL
1 mM 1.87 mL 9.37 mL 18.74 mL
5 mM 0.37 mL 1.87 mL 3.75 mL

*The above data is based on the productmolecular weight 533.6 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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