TC-MCH 7c is a selective antagonist of the melanin-concentrating hormone receptor 1 (MCH1R), featuring a phenylpyridone structure. This compound demonstrates high potency with an IC50 of 5.6 nM for human MCH1R, alongside Kis of 3.4 nM and 3.0 nM for human and mouse MCH1R, respectively. TC-MCH 7c is designed for oral administration and effectively penetrates the brain, making it a valuable tool for research in neurological disorders and metabolic regulation.
TC-MCH 7c is a selective antagonist of the melanin-concentrating hormone receptor 1 (MCH1R), featuring a phenylpyridone structure. This compound demonstrates high potency with an IC50 of 5.6 nM for human MCH1R, alongside Kis of 3.4 nM and 3.0 nM for human and mouse MCH1R, respectively. TC-MCH 7c is designed for oral administration and effectively penetrates the brain, making it a valuable tool for research in neurological disorders and metabolic regulation.
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