TD-6301 is a potent antagonist of the M2 and M4 muscarinic receptors, demonstrating high selectivity and strong affinity for the human M2 receptor (Ki = 0.36 nM). This compound effectively inhibits volume-induced bladder contractions (ID50 = 0.075 mg/kg), making it a valuable tool in the study of overactive bladder conditions. Its specificity for bladder tissues presents opportunities for targeted therapeutic research in urology and related fields.
TD-6301 is a potent antagonist of the M2 and M4 muscarinic receptors, demonstrating high selectivity and strong affinity for the human M2 receptor (Ki = 0.36 nM). This compound effectively inhibits volume-induced bladder contractions (ID50 = 0.075 mg/kg), making it a valuable tool in the study of overactive bladder conditions. Its specificity for bladder tissues presents opportunities for targeted therapeutic research in urology and related fields.
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