Tenalisib (RP6530)

Catalog No.: A16799

dual PI3Kδ/γ inhibitor

Tenalisib (RP6530)

Tenalisib (RP6530) Chemical Structure

CAS NO. 1639417-53-0

Tenalisib, also known as RP6530, is a potent and selective dual PI3Kδ/γ inhibitor that inhibited growth of B-cell lymphoma cell lines with a concomitant reduction in the downstream biomarker, pAKT.

Availability: In stock

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2 mg
$100.00
5 mg
$180.00
25 mg
$500.00
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Biological Activity

Tenalisib, also known as RP6530, is a potent and selective dual PI3Kδ/γ inhibitor that inhibited growth of B-cell lymphoma cell lines with a concomitant reduction in the downstream biomarker, pAKT.
In vitro DMSO 74 mg/mL (178.13 mM)
Water Insoluble
Ethanol 74 mg/mL (178.13 mM)
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 24.07 mL 120.36 mL 240.71 mL
0.5 mM 4.81 mL 24.07 mL 48.14 mL
1 mM 2.41 mL 12.04 mL 24.07 mL
5 mM 0.48 mL 2.41 mL 4.81 mL

*The above data is based on the productmolecular weight 415.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A16799
Actions Inhibitor
CAS No. 1639417-53-0
Formula C23H18FN5O2
M. Wt 415.43
Solubility DMSO
Purity >98%
Synonyms RP-6530, RP 6530
SMILES O=C1C(C2=CC=CC(F)=C2)=C([[email protected]@H](NC3=C4NC=NC4=NC=N3)CC)OC5=C1C=CC=C5
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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