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Tiplaxtinin (PAI-039)


PAI-1 inhbitor

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Catalog No. A14190

Availability:Stock in USAIn stock

Product Name Catalog No. Price Qty
Tiplaxtinin 5mg A14190-5

Regular Price: €71.25

Special Price: €64.13

Tiplaxtinin 10mg A14190-10

Regular Price: €80.75

Special Price: €72.68

Tiplaxtinin 25mg A14190-25

Regular Price: €190.00

Special Price: €171.00

Products are for laboratory research use only. Not for human use. We do not sell to patients.

Quick Overview

Tiplaxtinin is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 μM.

Tiplaxtinin (PAI-039)

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Publications citing Adooq Products
Tiplaxtinin (PAI-039) Citations (1)
  • Saijo A,et al. Bone marrow-derived fibrocytes promote stem cell-like properties of lung cancer cells, Cancer Lett, 2018, May 1;421:17-27 29448000

Chemical Information

Catalog Num A14190
Actions Inhibitor
M. Wt 439.3833
Formula C24H16F3NO4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 393105-53-8
Synonyms PAI-039
SMILES code C1=CC=C(C=C1)CN2C=C(C3=C2C=CC(=C3)C4=CC=C(C=C4)OC(F)(F)F)C(=O)C(=O)O
Chemical Name {1-benzyl-5-[4-(trifluoromethoxy)phenyl]-1H-indol-3-yl}(oxo)acetic acid

Biological Activity

Tiplaxtinin is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 μM.
2.7 μM

Preparing Stock Solutions

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.76 mL 113.8 mL 227.59mL
0.5 mM 4.55 mL 22.76 mL 45.52 mL
1 mM 2.28 mL 11.38 mL 22.76 mL
5 mM 0.46 mL 2.28 mL 4.55 mL

*The above data is based on the productmolecular weight 439.3833. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

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