Tiplaxtinin (PAI-039)

Catalog No.: A14190

PAI-1 inhbitor

Tiplaxtinin (PAI-039)

Tiplaxtinin (PAI-039) Chemical Structure

CAS NO. 393105-53-8

Tiplaxtinin is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 μM.

Availability: In stock

Package Price Qty
5 mg
$75.00
10 mg
$85.00
25 mg
$200.00
Custom Size Get quote

Free Overnight Delivery on orders over $500

Next day delivery by 10:00 a.m. Order now.

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Saijo A, .et al. Bone marrow-derived fibrocytes promote stem cell-like properties of lung cancer cells, Cancer Lett, 2018, May 1;421:17-27 PMID: 29448000

Biological Activity

Tiplaxtinin is a selective and orally efficacious inhibitor of plasminogen activator inhibitor-1 (PAI-1) with IC50 of 2.7 μM.
Targets
PAI-1
2.7 μM
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 22.76 mL 113.8 mL 227.59 mL
0.5 mM 4.55 mL 22.76 mL 45.52 mL
1 mM 2.28 mL 11.38 mL 22.76 mL
5 mM 0.46 mL 2.28 mL 4.55 mL

*The above data is based on the productmolecular weight 439.3833. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14190
Actions Inhibitor
M. Wt 439.3833
Formula C24H16F3NO4
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 393105-53-8
Synonyms PAI-039
SMILES C1=CC=C(C=C1)CN2C=C(C3=C2C=CC(=C3)C4=CC=C(C=C4)OC(F)(F)F)C(=O)C(=O)O

Product Tags

Product Tags

Other people marked this product with these tags:

Use spaces to separate tags. Use single quotes (') for phrases.

Product Questions

Product Questions

No Questions
Keywords:buy Tiplaxtinin (PAI-039) | Tiplaxtinin (PAI-039) Supplier | purchase | cost | manufacturer | order | distributor | buy 393105-53-8| 393105-53-8 Supplier | purchase 393105-53-8 | 393105-53-8 cost | 393105-53-8 manufacturer | order 393105-53-8 | 393105-53-8 distributor
Rewards