TOK-001 (Galeterone)

Catalog No.: A11138

CYP17 inhibitor

TOK-001 (Galeterone)

TOK-001 (Galeterone) Chemical Structure

CAS NO. 851983-85-2

TOK-001 (Galeterone) is both an androgen receptor antagonist and CYP17A1 inhibitor.

Availability: In stock

Package Price Qty
5 mg

Regular Price: $100.00

Special Price $90.00

10 mg

Regular Price: $180.00

Special Price $162.00

50 mg

Regular Price: $540.00

Special Price $486.00

100 mg

Regular Price: $850.00

Special Price $765.00

10mM * 1mL in DMSO

Regular Price: $110.00

Special Price $99.00

Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Biological Activity

TOK-001 (Galeterone) is both an androgen receptor antagonist and CYP17A1 inhibitor.
Targets
CYP17 Androgen Receptor
300 nM384 nM
In vitro (25°C) DMSO 24 mg/mL (61.76 mM)
Water <1 mg/mL (<1 mM)
Ethanol 40 mg/mL (102.94 mM)
In vivo 0.5% hydroxyethyl cellulose 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 25.75 mL 128.77 mL 257.53 mL
0.5 mM 5.15 mL 25.75 mL 51.51 mL
1 mM 2.58 mL 12.88 mL 25.75 mL
5 mM 0.52 mL 2.58 mL 5.15 mL

*The above data is based on the productmolecular weight 388.3 . Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Chemical Properties

Catalog Num A11138
Actions Inhibitor
M. Wt 388.3
Formula C26H32N2O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 851983-85-2
Synonyms VN/124-1
SMILES C[[email protected]]12CC[[email protected]@H](CC1=CC[[email protected]@H]3[[email protected]@H]2CC[[email protected]]4([[email protected]]3CC=C4N5C=NC6=CC=CC=C65)C)O

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