Fig. 1 · Structure
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TP-16
EP4 Antagonist
TP-16 is a selective antagonist of the EP4 receptor, demonstrating an IC50 value of 2.1 nM. This compound effectively inhibits EP4-mediated signaling pathways, making it a valuable tool for investigating the role of EP4 in various physiological and pathological processes. TP-16 is particularly relevant for research in inflammation, pain, and cancer biology, providing insights into therapeutic interventions targeting the prostaglandin receptor system.
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Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Antagonist |
| CAS Number | 2332972-26-4 |
| Applications | EP4 Antagonist |
| Formula | C24H22FNO4S |
| Molecular Weight | 439.50 |
| SMILES | C[C@@H](C1=CC=C(C=C1)C(O)=O)NC(C2=C(CC3=CC=C(C=C3)F)SC4=C2CCOC4)=O |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.