Vicriviroc Malate

Catalog No.: A10971

CCR5 antagonist

Vicriviroc Malate

Vicriviroc Malate Chemical Structure

CAS NO. 541503-81-5

Vicriviroc Malate is a second generation orally active CCR5 antagonist, which is also a potent inhibitor of HIV-1 entry into target cells, with a mean IC50 =0.46 nM and IC50 =1~10 nM to HIV isolates (n=52).

Availability: In stock

Package Price Qty
5 mg
$120.00
10 mg
$200.00
50 mg
$600.00
100 mg
$980.00
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Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.
  • Tomohiro Nabekura, .et al. Effects of Antiviral Drugs on Organic Anion Transport in Human Placental BeWo Cells, Antimicrob Agents Chemother, 2015, Dec; 59(12): 7666-7670 PMID: 26416870

Biological Activity

Vicriviroc Malate is a second generation orally active CCR5 antagonist, which is also a potent inhibitor of HIV-1 entry into target cells, with a mean IC50 =0.46 nM and IC50 =1~10 nM to HIV isolates (n=52).
In vitro DMSO 121 mg/mL (181.21 mM)
Water 34 mg/mL (50.92 mM)
Ethanol 121 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 14.98 mL 74.88 mL 149.77 mL
0.5 mM 3 mL 14.98 mL 29.95 mL
1 mM 1.5 mL 7.49 mL 14.98 mL
5 mM 0.3 mL 1.5 mL 3 mL

*The above data is based on the productmolecular weight 667.7. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A10971
Actions Antagonist
CAS No. 541503-81-5
Formula C28H38F3N5O2.C4H6O5
M. Wt 667.7
Purity >98%
SMILES C[[email protected]]1CN(CCN1[[email protected]@H](COC)C2=CC=C(C=C2)C(F)(F)F)C3(CCN(CC3)C(=O)C4=C(N=CN=C4C)C)C.C(C(C(=O)O)O)C(=O)O
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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