VS-5584

Catalog No.: A12480

PI3K/mTOR inhibitor

VS-5584

VS-5584 Chemical Structure

CAS NO. 1246560-33-7

VS-5584 is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.

Availability: In stock

Package Price Qty
10 mg

Regular Price: $120.00

Special Price $96.00

25 mg

Regular Price: $250.00

Special Price $200.00

50 mg

Regular Price: $400.00

Special Price $320.00

10mM * 1mL in DMSO
$95.00
Warning Products are for laboratory research use only. Not for human use. We do not sell to patients.

Details

VS-5584 is a novel and highly selective PI3K/mTOR kinase inhibitor for the treatment of cancer.
Targets
PI3Kα PI3Kδ PI3Kγ mTOR PI3Kβ
2.6 nM2.7 nM3.0 nM3.4 nM21 nM
In vitro (25°C) DMSO 71 mg/mL (200.33 mM)
Water <1 mg/mL (<1 mM)
Ethanol 3 mg/mL (8.46 mM)
In vivo 0.5% methylcellulose/0.2% Tween 80 30 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 28.22 mL 141.08 mL 282.16 mL
0.5 mM 5.64 mL 28.22 mL 56.43 mL
1 mM 2.82 mL 14.11 mL 28.22 mL
5 mM 0.56 mL 2.82 mL 5.64 mL

*The above data is based on the productmolecular weight 354.41. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Technical Details

Catalog Num A12480
Actions Inhibitor
M. Wt 354.41
Formula C17H22N8O
Solubility DMSO
Purity >98%
Storage at -20°C 3 years Powder
CAS No. 1246560-33-7
Synonyms SB2343, VS5584, SB-2343, SB 2343
SMILES CC1=NC2=C(N=C(N=C2N1C(C)C)N3CCOCC3)C4=CN=C(N=C4)N

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