Fig. 1 · Structure
Documents & Downloads
WAY-181187 oxalate
5-HT6 Agonist
WAY-181187 oxalate is a selective full agonist of the 5-HT6 receptor, exhibiting a binding affinity with a Ki of 2.2 nM and an effective concentration for half-maximal activation (EC50) of 6.6 nM. This compound engages 5-HT6 receptor-mediated signaling pathways, influencing cAMP, Fyn, and ERK1/2 kinase activity. It serves as a valuable tool for research into neuropharmacology and potential therapeutic applications targeting cognitive disorders.
In Stock
Free Aliquoting for Your Order
Tell us your preferred amount per vial. We’ll confirm the options.
Specifications
| Manufacturer | Adooq Bioscience |
|---|---|
| Actions | Agonist |
| CAS Number | 1883548-85-3 |
| Applications | 5-HT6 Agonist |
| Formula | C17H15ClN4O6S2 |
| Molecular Weight | 470.91 |
| Synonyms | SAX-187 oxalate |
| SMILES | OC(=O)C(O)=O.NCCc1cn(c2ccccc12)S(=O)(=O)c1c(Cl)nc2sccn12 |
Storage & Solubility
In Vitro Solubility
Reported Solubility
No reported solubility data are available for this product.
Preparing Stock Solutions
| Concentration | |
|---|---|
Values use four significant digits. Prepare to the final solution volume; this is not the volume of solvent to add.
Stock preparation is unavailable for this product molecular weight.
Calculated stock concentrations do not establish solvent solubility. Refer to the reported solubility data for experimental guidance.
Storage
Store powder at -20°C, keep desiccated.
In powder form, the chemical is stable for 36 months.
In solution, store at -20°C and use within 1 month to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.