Telaglenastat (CB-839)

Catalog No.: A14396
Glutaminase inhibitor

CB-839 an is orally bioavailable inhibitor of glutaminase, with potential antineoplastic activity. CB-839 (Telaglenastat) also inudces autophagy and has antitumor activity.

Grouped product items
Product Name Price Stock Qty
CB-839 5mg
Special Price $44.00 Regular Price $55.00
In stock
CB-839 10mg
Special Price $64.00 Regular Price $80.00
In stock
CB-839 25mg
Special Price $128.00 Regular Price $160.00
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Important Notice: For research use only. We do not sell to patients.

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Adooq Products cited in reputable paper
Adooq's Telaglenastat (CB-839) has been cited by 1 publications
  • Beatriz Giesen, .et al. , Pharmaceutics, 2021, Feb 23;13(2):295 PMID: 33672398
  • Biological Activity
    Discription

    CB-839 an is orally bioavailable inhibitor of glutaminase, with potential antineoplastic activity. CB-839 (Telaglenastat) also inudces autophagy and has antitumor activity.

    Targets
    Target Value
    Product Information
    Catalog Num A14396
    Formula C26H24F3N7O3S
    Molecular Weight 571.57
    CAS Number 1439399-58-2
    SMILES O=C(CC1=CC=CC(OC(F)(F)F)=C1)NC2=CC=C(CCCCC3=NN=C(NC(CC4=NC=CC=C4)=O)S3)N=N2
    Synonyms CB839, CB 839
    Storage

    Store lyophilized at -20ºC, keep desiccated.
    In lyophilized form, the chemical is stable for 36 months.
    In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

    Solubility
    In vitro (25°C) DMSO Warmed: 97 mg/mL (169.7 mM)
    Water Insoluble
    Ethanol Insoluble
    In vivo 5% DMSO+corn oil 2 mg/mL
    * <1 mg/ml means slightly soluble or insoluble.
    * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
    Preparing Stock Solutions
    Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
    0.1 mM 17.5 mL 87.48 mL 174.96 mL
    0.5 mM 3.5 mL 17.5 mL 34.99 mL
    1 mM 1.75 mL 8.75 mL 17.5 mL
    5 mM 0.35 mL 1.75 mL 3.5 mL
    Useful Calculator

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    Calculate the dilution required to prepare a stock solution.
    This equation is commonly abbreviated as: C1V1 = C2V2

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