CB-839

Catalog No.: A14396

Glutaminase inhibitor

CB-839

CB-839 Chemical Structure

CAS NO. 1439399-58-2

CB-839 an is orally bioavailable inhibitor of glutaminase, with potential antineoplastic activity.

Availability: In stock

Package Price Qty
5 mg
$55.00
10 mg
$80.00
25 mg
$160.00
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Biological Activity

CB-839 an is orally bioavailable inhibitor of glutaminase, with potential antineoplastic activity.
Targets
glutaminase
24 nM
In vitro (25°C) DMSO Warmed: 97 mg/mL (169.7 mM)
Water Insoluble
Ethanol Insoluble
In vivo 5% DMSO+corn oil 2 mg/mL
* <1 mg/ml means slightly soluble or insoluble.
* Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations.
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
0.1 mM 17.5 mL 87.48 mL 174.96 mL
0.5 mM 3.5 mL 17.5 mL 34.99 mL
1 mM 1.75 mL 8.75 mL 17.5 mL
5 mM 0.35 mL 1.75 mL 3.5 mL

*The above data is based on the productmolecular weight 571.57. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Catalog Num A14396
Actions Inhibitor
CAS No. 1439399-58-2
Formula C26H24F3N7O3S
M. Wt 571.57
Solubility DMSO
Purity >98%
Synonyms CB839, CB 839
SMILES O=C(CC1=CC=CC(OC(F)(F)F)=C1)NC2=CC=C(CCCCC3=NN=C(NC(CC4=NC=CC=C4)=O)S3)N=N2
Storage

Store lyophilized at -20ºC, keep desiccated.
In lyophilized form, the chemical is stable for 36 months.
In solution, store at -20ºC and use within 3 months to prevent loss of potency. Aliquot to avoid multiple freeze/thaw cycles.

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