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- Leo Shen, .et al. A forward genetic screen identifies modifiers of rocaglate responsiveness, Sci Rep, 2021, Sep 16;11(1):18516 PMID: 34531456
Biological Activity
Elacridaris a prototypical BCRP inhibitor which inhibits the Bcrp1-mediated transport.
Targets
| P-gp | BCRP | |||
| In vitro (25°C) | DMSO | Warmed: 7 mg/mL (12.42 mM) | |
| Water | Insoluble | ||
| Ethanol | Insoluble | ||
| In vivo | 4% DMSO+30% PEG 300+5% Tween 80+ddH2O | 1 mg/mL | |
|
* <1 mg/ml means slightly soluble or insoluble. * Please note that Adooq tests the solubility of all compounds in-house, and the actual solubility may differ slightly from published values. This is normal and is due to slight batch-to-batch variations. |
|||
| Concentration / Solvent Volume / Mass | 1 mg | 5 mg | 10 mg |
|---|---|---|---|
| 0.1 mM | 17.74 mL | 88.71 mL | 177.42 mL |
| 0.5 mM | 3.55 mL | 17.74 mL | 35.48 mL |
| 1 mM | 1.77 mL | 8.87 mL | 17.74 mL |
| 5 mM | 0.35 mL | 1.77 mL | 3.55 mL |
*The above data is based on the productmolecular weight 563.64. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
| Catalog Num | A12324 |
|---|---|
| Actions | Inhibitor |
| CAS No. | 143664-11-3 |
| Formula | C34H33N3O5 |
| M. Wt | 563.64 |
| Purity | >98% |
| SMILES | COC1=CC=CC2=C1NC3=C(C2=O)C=CC=C3C(=O)NC4=CC=C(C=C4)CCN5CCC6=CC(=C(C=C6C5)OC)OC |
| Storage | Store lyophilized at -20ºC, keep desiccated. |
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