Name: YHO-13351 free base
SKU: A21568
Price: 90 USD
Rating: 5 (288 reviews)

Catalog No.

Product Name

Application

Product Information

Product Citation

A11475

Ko-143

BCRP inhibitor

Ko 143 is potent and selective inhibitor of breast cancer resistance protein multidrug transporter (BCRP) with an EC90 value of 26 nM.

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A12324

Elacridar (GF120918)

P-gp & BCRP inhibitor

Elacridaris a prototypical BCRP inhibitor which inhibits the Bcrp1-mediated transport.

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- Leo Shen, .et al. , Sci Rep, 2021, Sep 16;11(1):18516 PMID: 34531456
A16195

KS-176

BCRP inhibitor

KS-176 is a potent and selective inhibitor of the breast cancer resistance protein (BCRP) multidrug transporter (IC50 values are 0.59 and 1.39 uM in Pheo A and Hoechst 33342 assays respectively).

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A17127

YHO-13177

BCRP/ABCG2 inhibitor

YHO-13177 is a potent and specific inhibitor of breast cancer resistance protein (BCRP/ABCG2).

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A18393

FD 12-9

P-gp/BCRP dual inhibitor

FD 12-9 is a flavonoid dimer, acts as a dual inhibitor of P-gp and BCRP, with EC50s of 285 nM and 0.9 nM, respectively. Anti-glioblastoma activity.

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A20298

ML230

ABCG2 inhibitor

ML230 (CID44640177; SID 88095709) is a selective inhibitor of ATP-binding cassette (ABC) transporter ABCG2, and 36-fold selective for ABCG2 over ABCB1 with EC50s values of 0.13 μM and 4.65 μM, respectively.

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A20588

(S)-ML753286

BCRP inhibitor

(S)-ML753286 is a breast cancer resistance protein (BCRP) inhibitor with an IC50 of 0.6 μM on BCRP efflux transporter.

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A21568

YHO-13351 free base

BCRP inhibitor

YHO-13351 (free base) is the water-soluble prodrug of YHO-13177, which is a potent and specific inhibitor of BCRP.

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BCRP